SCHEMBL8096944

SCHEMBL8096944

CCOC(=O)CNC(=O)Oc1ncc(C(=O)NS(=O)(=O)c2ccc(C(=O)N(CC)CC)cc2)cc1OC

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.39
LMNA P02545 1/20 0.39
HPGD P15428 1/20 0.39
HTT P42858 1/20 0.39
ABL1 P00519 1/20 0.39
RIN1 Q13671 1/20 0.39
P4HTM Q9NXG6 1/20 0.38
CYP1A2 P05177 1/20 0.37
HSP90AA1 P07900 1/20 0.37
HSP90AB1 P08238 1/20 0.37
BLM P54132 1/20 0.37
PTGS2 P35354 1/20 0.37
EGFR P00533 3/20 0.36
NAMPT P43490 1/20 0.36
LRRK2 Q5S007 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
SCN9A Q15858 2/20 0.34
L3MBTL1 Q9Y468 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8099328 0.94 P4HTM (0.37) SMN1; SMN2P4HTMPTGS2EGFRMEN1
SCHEMBL8767162 0.91 LMNA (0.40) SMN1; SMN2LMNAHPGDHTTABL1
SCHEMBL8099449 0.91 LMNA (0.37) SMN1; SMN2LMNAHPGDHTTPTGS2
SCHEMBL8106135 0.90 LMNA (0.40) SMN1; SMN2LMNAHPGDHTTP4HTM
SCHEMBL8097664 0.90 ABL1 (0.37) SMN1; SMN2LMNAHPGDHTTABL1
SCHEMBL8104048 0.88 PTGS2 (0.44) SMN1; SMN2P4HTMPTGS2EGFRKMT2A
SCHEMBL8875475 0.87 P4HTM (0.39) SMN1; SMN2LMNAHPGDHTTABL1
SCHEMBL8768258 0.84 CA1 (0.39) P4HTMPTGS2EGFRSCN9A
SCHEMBL8768279 0.84 LMNA (0.42) SMN1; SMN2LMNAHPGDHTTCYP1A2
SCHEMBL8767144 0.81 LMNA (0.38) SMN1; SMN2LMNAHPGDHTTP4HTM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0673932-B1 Sulfonamidocarbonyl-pyridine-2-carboxamides as well as their pyridine-N-oxides, process for their preparation and their use as medicaments HOECHST AG (DE) 2000-06-07 EP disclosed
EP-0673932-A1 Sulfonamidocarbonyl-pyridine-2-carboxamides as well as their pyridine-N-oxides, process for their preparation and their use as medicaments HOECHST AKTIENGESELLSCHAFT (DE) 1995-09-27 EP disclosed