SCHEMBL8769578

SCHEMBL8769578

CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](Cc1ccccc1)[C@@H](O)C(=O)NCc1ccncc1

nearest known ligand 0.59

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CTSD P07339 3/20 0.59
BACE1 P56817 10/20 0.57
CTSB P07858 2/20 0.56
CTSL P07711 1/20 0.56
CTSS P25774 1/20 0.56
MEN1 O00255 2/20 0.54
KMT2A Q03164 2/20 0.54
LMNA P02545 1/20 0.54
PSMB1 P20618 1/20 0.53
ALDH1A1 P00352 1/20 0.50
CYP3A4 P08684 1/20 0.50
CTSK P43235 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8769560 0.94 CTSD (0.65) CTSDBACE1CTSBCTSLCTSS
SCHEMBL8769497 0.88 REN (0.59) CTSDCTSBCTSLCTSSMEN1
SCHEMBL8770005 0.86 CTSB (0.60) CTSDCTSBCTSLCTSSMEN1
SCHEMBL8769526 0.85 CTSL (0.63) CTSDCTSBCTSLCTSSMEN1
SCHEMBL16463050 0.84 PSMB1 (0.57) CTSDBACE1PSMB1ALDH1A1CYP3A4
SCHEMBL16463052 0.84 PSMB1 (0.57) CTSDBACE1PSMB1ALDH1A1CYP3A4
SCHEMBL16463049 0.84 PSMB1 (0.57) CTSDBACE1PSMB1ALDH1A1CYP3A4
SCHEMBL16463054 0.84 PSMB1 (0.57) CTSDBACE1PSMB1ALDH1A1CYP3A4
SCHEMBL7269133 0.83 CTSB (0.65) CTSDCTSBCTSLCTSSMEN1
SCHEMBL6448856 0.83 CTSB (0.65) CTSDCTSBCTSLCTSSMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0793673-A1 ALPHA-KETOAMIDE DERIVATIVES AS CATHEPSIN L INHIBITOR Takeda Chemical Industries, Ltd. (JP) 1997-09-10 EP disclosed
WO-1996016079-A2 ALPHA-KETOAMIDE DERIVATIVES AS CATHEPSIN L INHIBITOR TAKEDA CHEMICAL INDUSTRIES, LTD (JP) 1996-05-30 WO disclosed