SCHEMBL8772949

SCHEMBL8772949

O=C(c1cc(C(F)(F)F)ccc1O)c1ncccc1O

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR7 Q9NYK1 6/20 0.56
KCNMA1 Q12791 1/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
P2RX1 P51575 2/20 0.41
CES2 O00748 1/20 0.41
CNR2 P34972 2/20 0.40
NPC1 O15118 1/20 0.40
CRHBP P24387 1/20 0.40
RAB9A P51151 1/20 0.40
CRHR2 Q13324 1/20 0.40
GMNN O75496 1/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
TTR P02766 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
PKM P14618 1/20 0.40
NFKB1 P19838 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8712176 0.79 GSTA1 (0.63) TLR7MEN1KMT2ACES2NPC1
SCHEMBL8709808 0.78 CSNK2A1 (0.50) MEN1KMT2ANPC1RAB9AALDH1A1
SCHEMBL8654976 0.77 FTO (0.45) TLR7ALDH1A1LMNACYP3A4COMT
SCHEMBL8709073 0.76 KDM4E (0.50) TLR7MEN1KMT2AALDH1A1LMNA
SCHEMBL8714018 0.75 KDM4E (0.43) TLR7MEN1KMT2ANPC1RAB9A
SCHEMBL8709612 0.75 TLR7 (0.42) TLR7KCNMA1KMT2AALDH1A1LMNA
SCHEMBL8709608 0.75 TLR7 (0.42) TLR7KCNMA1KMT2AALDH1A1LMNA
SCHEMBL8711999 0.74 TRPA1 (0.42) TLR7NPC1RAB9ACYP1A2CYP2C9
SCHEMBL8709049 0.74 MAPT (0.53) MEN1KMT2ANPC1RAB9AALDH1A1
SCHEMBL5992479 0.74 CNR2 (0.55) MEN1KMT2AP2RX1CES2CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0623597-B1 Pyridine derivatives, with potassium channel opening activity TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1997-10-22 EP disclosed
EP-0623597-A1 Pyridine derivatives, with potassium channel opening activity Takeda Chemical Industries, Ltd. (JP) 1994-11-09 EP disclosed