SCHEMBL8709808

SCHEMBL8709808

Cc1ccc(O)c(C(=O)c2ncccc2O)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CSNK2A1 P68400 1/20 0.50
COMT P21964 1/20 0.46
HPGD P15428 6/20 0.45
HTT P42858 4/20 0.45
MAPT P10636 3/20 0.45
SPR P35270 2/20 0.45
GRM5 P41594 1/20 0.43
KDM4E B2RXH2 3/20 0.42
L3MBTL1 Q9Y468 4/20 0.42
LMNA P02545 4/20 0.42
ALDH1A1 P00352 3/20 0.41
GSTA1 P08263 1/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
RAB9A P51151 1/20 0.41
KDR P35968 1/20 0.41
MAPK1 P28482 3/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
TP53 P04637 1/20 0.41
EGLN2 Q96KS0 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8712176 0.83 GSTA1 (0.63) HPGDMAPTSPRKDM4EALDH1A1
SCHEMBL8709049 0.81 MAPT (0.53) HPGDHTTMAPTSPRKDM4E
SCHEMBL8711999 0.81 TRPA1 (0.42) HPGDMAPTSPRKDM4EGSTA1
SCHEMBL8654976 0.80 FTO (0.45) COMTMAPTSPRKDM4EL3MBTL1
SCHEMBL8709073 0.80 KDM4E (0.50) HPGDHTTMAPTSPRKDM4E
SCHEMBL8714018 0.79 KDM4E (0.43) HPGDMAPTSPRKDM4EL3MBTL1
SCHEMBL8709727 0.79 KDM5A (0.44) HPGDMAPTKDM4EALDH1A1MEN1
SCHEMBL8772949 0.78 TLR7 (0.56) COMTLMNAALDH1A1GSTA1MEN1
SCHEMBL27699633 0.77 FTO (0.55) COMTMAPTSPRKDM4EL3MBTL1
SCHEMBL11500852 0.77 CSNK2A1 (0.72) CSNK2A1HPGDHTTMAPTSPR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5716971-A FOR TREATMENT OF ANGINA PECTORIS AND HYPERTENSION TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-10 US disclosed
EP-0623597-B1 Pyridine derivatives, with potassium channel opening activity TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1997-10-22 EP disclosed
EP-0623597-A1 Pyridine derivatives, with potassium channel opening activity Takeda Chemical Industries, Ltd. (JP) 1994-11-09 EP disclosed