SCHEMBL8775147

SCHEMBL8775147

CCCc1ccc(CCc2cnc(F)c(F)c2)cc1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.47
RAB9A P51151 3/20 0.47
TP53 P04637 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
PKM P14618 1/20 0.47
HSD17B10 Q99714 1/20 0.47
LPL P06858 1/20 0.36
LIPG Q9Y5X9 1/20 0.36
CNR1 P21554 1/20 0.35
CNR2 P34972 1/20 0.35
MAPT P10636 1/20 0.35
GFER P55789 1/20 0.35
PDGFRB P09619 1/20 0.35
PDGFRA P16234 1/20 0.35
CA2 P00918 1/20 0.34
GPR84 Q9NQS5 1/20 0.34
HTR2A P28223 1/20 0.34
KCNH2 Q12809 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8774337 0.95 RAB9A (0.50) NPC1RAB9ATP53SMN1; SMN2PKM
SCHEMBL8774481 0.90 NFKB1 (0.44) NPC1RAB9ATP53SMN1; SMN2PKM
SCHEMBL8774752 0.89 TAAR1 (0.44) NPC1RAB9ATP53SMN1; SMN2PKM
SCHEMBL8774239 0.87 HTR2A (0.50) NPC1RAB9ATP53SMN1; SMN2HSD17B10
SCHEMBL8774784 0.85 RAB9A (0.46) NPC1RAB9ATP53SMN1; SMN2PKM
SCHEMBL8774132 0.85 NPC1 (0.40) NPC1RAB9ATP53SMN1; SMN2PKM
SCHEMBL8774178 0.84 CYP3A4 (0.43) NPC1RAB9ASMN1; SMN2PKMHSD17B10
SCHEMBL8774406 0.84 RARB (0.50) NPC1RAB9ASMN1; SMN2HSD17B10MAPT
SCHEMBL8774716 0.84 LMNA (0.47) NPC1RAB9ASMN1; SMN2HSD17B10MAPT
SCHEMBL8774669 0.83 NQO1 (0.44) RAB9ATP53SMN1; SMN2MAPTPDGFRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0519370-B1 Heterocyclic derivatives MERCK PATENT GMBH (DE) 1997-11-05 EP disclosed
EP-0519370-A2 Heterocyclic derivatives MERCK PATENT GmbH (DE) 1992-12-23 EP disclosed