SCHEMBL8774858

SCHEMBL8774858

CCCCCOc1ccc(CCc2cnc(F)c(F)c2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.44
USP2 O75604 1/20 0.44
ALDH1A1 P00352 1/20 0.44
LMNA P02545 1/20 0.44
CYP3A4 P08684 1/20 0.44
MAPK1 P28482 1/20 0.44
CASP1 P29466 1/20 0.44
KMT2A Q03164 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
SLCO1B3 Q9NPD5 1/20 0.44
SLCO1B1 Q9Y6L6 1/20 0.44
RAB9A P51151 2/20 0.43
MAPT P10636 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
NR5A1 Q13285 1/20 0.43
LTA4H P09960 2/20 0.42
S1PR4 O95977 2/20 0.41
S1PR1 P21453 2/20 0.41
S1PR3 Q99500 2/20 0.41
S1PR5 Q9H228 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8774178 0.97 CYP3A4 (0.43) MEN1USP2ALDH1A1LMNACYP3A4
SCHEMBL8774716 0.92 LMNA (0.47) ALDH1A1LMNASMN1; SMN2RAB9AMAPT
SCHEMBL8774239 0.85 HTR2A (0.50) MEN1USP2ALDH1A1LMNACYP3A4
SCHEMBL8774669 0.85 NQO1 (0.44) ALDH1A1LMNASMN1; SMN2RAB9AMAPT
SCHEMBL8774481 0.85 NFKB1 (0.44) MEN1USP2ALDH1A1LMNACYP3A4
SCHEMBL8774406 0.83 RARB (0.50) MEN1USP2ALDH1A1MAPK1KMT2A
SCHEMBL8775147 0.82 NPC1 (0.47) SMN1; SMN2RAB9AMAPTNPC1
SCHEMBL8774784 0.81 RAB9A (0.46) MEN1USP2ALDH1A1LMNACYP3A4
SCHEMBL9160679 0.81 MAPT (0.49) MEN1USP2ALDH1A1LMNACYP3A4
SCHEMBL8774813 0.81 MEN1 (0.42) MEN1USP2ALDH1A1LMNACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0519370-B1 Heterocyclic derivatives MERCK PATENT GMBH (DE) 1997-11-05 EP disclosed
EP-0519370-A2 Heterocyclic derivatives MERCK PATENT GmbH (DE) 1992-12-23 EP disclosed