SCHEMBL8774882

SCHEMBL8774882

CCCc1ccc(-c2cnc(Cl)c(Cl)c2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.41
SMN1; SMN2 Q16637 5/20 0.41
NPC1 O15118 4/20 0.41
TP53 P04637 2/20 0.41
HSD17B10 Q99714 2/20 0.41
PKM P14618 1/20 0.41
MAP4K4 O95819 1/20 0.40
AKR1C2 P52895 1/20 0.40
AKR1C1 Q04828 1/20 0.40
MAPT P10636 2/20 0.40
GFER P55789 1/20 0.40
MCL1 Q07820 1/20 0.39
PTGS2 P35354 1/20 0.39
ALDH1A1 P00352 5/20 0.38
NPSR1 Q6W5P4 2/20 0.38
KDM4E B2RXH2 3/20 0.37
GAA P10253 3/20 0.37
NISCH Q9Y2I1 1/20 0.37
POLB P06746 1/20 0.37
CTDSP1 Q9GZU7 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8774724 0.90 AKR1C2 (0.50) RAB9ASMN1; SMN2NPC1TP53HSD17B10
SCHEMBL8774115 0.89 RAB9A (0.49) RAB9ASMN1; SMN2NPC1HSD17B10AKR1C2
SCHEMBL8774222 0.88 MAPT (0.51) RAB9ASMN1; SMN2NPC1HSD17B10AKR1C2
SCHEMBL8774963 0.88 MAPT (0.51) RAB9ASMN1; SMN2NPC1HSD17B10AKR1C2
SCHEMBL8774839 0.86 EGLN1 (0.45) RAB9ASMN1; SMN2NPC1TP53MAP4K4
SCHEMBL8774671 0.85 NPC1 (0.42) RAB9ASMN1; SMN2NPC1TP53HSD17B10
SCHEMBL8774683 0.83 RAB9A (0.40) RAB9ASMN1; SMN2NPC1TP53HSD17B10
SCHEMBL8774299 0.82 GPR84 (0.36) RAB9ASMN1; SMN2NPC1MAP4K4AKR1C2
SCHEMBL8774303 0.82 GPR84 (0.36) RAB9ASMN1; SMN2NPC1MAP4K4AKR1C2
SCHEMBL8774328 0.80 GPR84 (0.38) RAB9ASMN1; SMN2NPC1HSD17B10MAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0519370-B1 Heterocyclic derivatives MERCK PATENT GMBH (DE) 1997-11-05 EP disclosed
EP-0519370-A2 Heterocyclic derivatives MERCK PATENT GmbH (DE) 1992-12-23 EP disclosed