SCHEMBL8779283

SCHEMBL8779283

CC(C)Oc1ccnc(OC(=O)NC(=O)CN)c1O

nearest known ligand 0.35

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.35
ACHE P22303 1/20 0.35
GRIN3B O60391 1/20 0.35
GRIN1 Q05586 1/20 0.35
GRIN2C Q14957 1/20 0.35
IRAK4 Q9NWZ3 18/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8779122 0.87 MAPT (0.33) ALDH1A1
SCHEMBL8779326 0.85 SMN1; SMN2 (0.39)
SCHEMBL8779253 0.85 HTT (0.39)
SCHEMBL8779267 0.84 ALDH1A1 (0.36) ALDH1A1ACHEGRIN3BGRIN1GRIN2C
SCHEMBL8779308 0.84 ALDH1A1 (0.36) ALDH1A1ACHEGRIN3BGRIN1GRIN2C
SCHEMBL8779273 0.83 IKBKB (0.38) ALDH1A1
SCHEMBL8779284 0.82 NFKB1 (0.32)
SCHEMBL8779138 0.82 SMN1; SMN2 (0.39)
SCHEMBL8779241 0.81 LMNA (0.40)
SCHEMBL8779087 0.81 IKBKB (0.34) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0661269-B1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AG (DE) 1997-03-26 EP disclosed
EP-0661269-A1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AKTIENGESELLSCHAFT (DE) 1995-07-05 EP disclosed