SCHEMBL878683

SCHEMBL878683

CC(C)(F)CNC1CCc2ccc(C(=O)O)cc21

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAOA P21397 3/20 0.42
MAOB P27338 3/20 0.42
ACHE P22303 12/20 0.41
DRD3 P35462 1/20 0.41
WDR5 P61964 1/20 0.38
BCHE P06276 1/20 0.38
TBXA2R P21731 1/20 0.38
PDE4A P27815 1/20 0.37
PDE4B Q07343 1/20 0.37
PDE4C Q08493 1/20 0.37
PDE4D Q08499 1/20 0.37
ALDH1A1 P00352 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL484566 0.90 MAOA (0.41) MAOAMAOBACHEDRD3WDR5
SCHEMBL784661 0.83 ACHE (0.57) MAOAMAOBACHEDRD3BCHE
SCHEMBL784930 0.81 WDR5 (0.43) ACHEDRD3WDR5PDE4APDE4B
SCHEMBL784931 0.81 WDR5 (0.43) ACHEDRD3WDR5PDE4APDE4B
SCHEMBL784108 0.81 MAOA (0.45) MAOAMAOBACHEDRD3BCHE
SCHEMBL484717 0.79 CHRNB2 (0.46) MAOAMAOBACHEBCHE
SCHEMBL484719 0.79 CHRNB2 (0.46) MAOAMAOBACHEBCHE
SCHEMBL484852 0.78 ACHE (0.54) MAOAMAOBACHEDRD3PDE4A
SCHEMBL484623 0.78 HTR1A (0.43) DRD3WDR5TBXA2RPDE4APDE4B
SCHEMBL784704 0.78 TAS1R3 (0.45) ACHEDRD3WDR5TBXA2RPDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2619178-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2013-07-31 EP disclosed
WO-2012038081-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2012-03-29 WO disclosed