SCHEMBL8799072

SCHEMBL8799072

Cn1cc(C(N)=O)c(Cl)n1

nearest known ligand 0.63

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.41
ADORA1 P30542 2/20 0.41
ADRA1D P25100 1/20 0.37
POLB P06746 2/20 0.37
LMNA P02545 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
PARP1 P09874 5/20 0.36
PARP2 Q9UGN5 2/20 0.36
PARP3 Q9Y6F1 2/20 0.36
IRAK4 Q9NWZ3 3/20 0.35
MGLL Q99685 1/20 0.35
NNMT P40261 1/20 0.35
TSHR P16473 1/20 0.35
GAA P10253 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6249101 0.82 ALKBH1 (0.41) ADORA2AADORA1POLBLMNAL3MBTL1
SCHEMBL27497366 0.82 ADORA2A (0.38) ADORA2AADORA1POLBLMNAL3MBTL1
SCHEMBL15307202 0.82 LMNA (0.41) ADORA2AADORA1POLBLMNAL3MBTL1
SCHEMBL29002489 0.79 ADORA2A (0.42) ADORA2AADORA1L3MBTL1PARP1PARP2
SCHEMBL174293 0.78 ADORA2A (0.45) ADORA2AADORA1L3MBTL1GAA
SCHEMBL1224892 0.78 GAA (0.50) ADORA2AADORA1POLBNNMTGAA
SCHEMBL1833232 0.78 ADORA2A (0.49) ADORA2AADORA1LMNAL3MBTL1IRAK4
SCHEMBL7979529 0.77 GAA (0.46) ADORA2APOLBLMNAL3MBTL1TSHR
SCHEMBL15307174 0.77 ALDH1A1 (0.39) ADORA2AADORA1POLBLMNAMGLL
SCHEMBL20524576 0.77 GAA (0.39) ADORA2AADORA1POLBIRAK4NNMT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025119372-A2 MRGPRX2 ANTAGONIST AND USE THEREOF 武汉人福创新药物研发中心有限公司 2025-06-12 WO disclosed
CN-120118069-A MRGPRX2 antagonists and uses 武汉人福创新药物研发中心有限公司 2025-06-10 CN disclosed
US-12240862-B2 Inhibitors of peptidylarginine deiminases GILEAD SCIENCES, INC. (US) 2025-03-04 US disclosed
WO-2023192901-A9 QUINOLINE DERIVATIVES AS MODULATORS OF MAS-RELATED G-PROTEIN RECEPTOR X2 AND RELATED PRODUCTS ESCIENT PHARMACEUTICALS, INC. (US) 2023-12-14 WO disclosed
WO-2023192901-A1 QUINOLINE DERIVATIVES AS MODULATORS OF MAS-RELATED G-PROTEIN RECEPTOR X2 AND RELATED PRODUCTS ESCIENT PHARMACEUTICALS, INC. (US) 2023-10-05 WO disclosed
CN-101291584-A Herbicide composition NISSAN CHEMICAL IND LTD (JP) 2008-10-22 CN disclosed
EP-0537423-B1 N-pyrazolyl-1,2,4-triazolo(1,5-c)pyrimidine-2-sulfonamide herbicides DOWELANCO (US) 1997-10-08 EP disclosed
CN-1033806-C Herbicidal composition DOWELANCO (US) 1997-01-15 CN disclosed
CN-1134223-A Method for controling needless plant DOWELANCO (US) 1996-10-30 CN disclosed
EP-0537423-A1 N-pyrazolyl-1,2,4-triazolo(1,5-c)pyrimidine-2-sulfonamide herbicides DowElanco (US) 1993-04-21 EP disclosed
US-5201938-A N-pyrazolyl-1,2,4-triazolo[1,5-c]pyrimidine-2-sulfonamide herbicides DOWELANCO (US) 1993-04-13 US disclosed
CN-1068824-A N-pyrazolyl-1, 2, 4-triazolo [1, 5-c ] pyrimidine-2-sulfonamides as herbicides DOWELANCO (US) 1993-02-10 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12240862-B2 Inhibitors of peptidylarginine deiminases PADI4, PADI2, PADI1 ADORA2A 2714/4885ADORA1 3747/4885ADRA1D 4385/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.