SCHEMBL8799600

SCHEMBL8799600

COc1ccccc1NC(=O)CC(CC(=O)OC(=O)CC(CC(=O)OC(=O)CC(CC(=O)Nc1ccccc1OC)c1ccc(Cl)c(Cl)c1)c1ccc(Cl)c(Cl)c1)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.48
HTT P42858 2/20 0.48
ALDH1A1 P00352 3/20 0.47
LMNA P02545 2/20 0.47
NPSR1 Q6W5P4 1/20 0.47
MAPT P10636 5/20 0.46
KDM4E B2RXH2 2/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
MAPK10 P53779 1/20 0.46
POLB P06746 2/20 0.45
GAA P10253 1/20 0.45
RECQL P46063 1/20 0.45
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
SLC6A2 P23975 1/20 0.43
SLC6A4 P31645 1/20 0.43
SLC6A3 Q01959 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8799599 0.96 FNTA (0.49) HPGDHTTALDH1A1LMNANPSR1
SCHEMBL7811262 0.90 FNTA (0.53) HPGDHTTALDH1A1LMNANPSR1
SCHEMBL8799604 0.77 FNTA (0.42) HPGDHTTALDH1A1LMNANPSR1
SCHEMBL692174 0.75 LMNA (0.49) HTTALDH1A1LMNAMAPTRAB9A
SCHEMBL28673750 0.73 ALDH1A1 (0.60) HPGDHTTALDH1A1LMNANPSR1
SCHEMBL8798403 0.73 PRKCZ (0.48) HTTALDH1A1LMNAMEN1KMT2A
SCHEMBL657182 0.73 PRKCZ (0.48) HTTALDH1A1LMNAMEN1KMT2A
SCHEMBL7812248 0.72 MTNR1A (0.49) HPGDHTT
SCHEMBL12268167 0.71 FNTA (0.47) HTTALDH1A1LMNAGAASLC6A3
SCHEMBL9311962 0.70 MEN1 (0.64) HPGDHTTALDH1A1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0773929-A1 PIPERIDINE DERIVATIVES AS NEUROKININ ANTAGONISTS SCHERING CORPORATION (US) 1997-05-21 EP disclosed
WO-1996039386-A1 PIPERIDINE DERIVATIVES AS NEUROKININ ANTAGONISTS SCHERING CORPORATION (US) 1996-12-12 WO disclosed