SCHEMBL8801508

SCHEMBL8801508

O=C1CCc2cccc(OCc3ccc(OCc4ccc5ccccc5n4)cc3)c2N1

nearest known ligand 0.51

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYSLTR1 Q9Y271 6/20 0.51
FFAR1 O14842 1/20 0.48
AKR1B1 P15121 1/20 0.48
CYSLTR2 Q9NS75 5/20 0.48
ALOX5 P09917 2/20 0.47
GPBAR1 Q8TDU6 1/20 0.47
PDE10A Q9Y233 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8801669 0.90 CYSLTR1 (0.54) CYSLTR1CYSLTR2ALOX5GPBAR1
SCHEMBL8800823 0.82 CYSLTR1 (0.48) CYSLTR1FFAR1AKR1B1CYSLTR2ALOX5
SCHEMBL8800332 0.80 CYSLTR1 (0.51) CYSLTR1FFAR1AKR1B1CYSLTR2ALOX5
SCHEMBL8801873 0.77 MAOB (0.58) CYSLTR1FFAR1AKR1B1CYSLTR2PDE10A
SCHEMBL6584872 0.75 DRD2 (0.48)
SCHEMBL10544473 0.75 CYSLTR1 (0.84) CYSLTR1FFAR1AKR1B1CYSLTR2ALOX5
SCHEMBL6586928 0.74 MAOA (0.45)
SCHEMBL8800538 0.74 CYSLTR1 (0.51) CYSLTR1CYSLTR2ALOX5GPBAR1
SCHEMBL9022146 0.73 GPBAR1 (0.66) CYSLTR1FFAR1AKR1B1CYSLTR2ALOX5
SCHEMBL8308890 0.73 DRD2 (0.49)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0799826-A1 Heteroaryl substituted phenylene derivatives, their preparation and their use as leukotriene receptor antagonists KOWA CO. LTD. (JP) 1997-10-08 EP disclosed