SCHEMBL8828332

SCHEMBL8828332

COc1ccc(CCN(C)CCCNC(=O)C/C=C/c2cccc(C#N)c2)cc1OC

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 3/20 0.47
TMEM97 Q5BJF2 3/20 0.47
SIGMAR1 Q99720 3/20 0.47
LMNA P02545 1/20 0.46
HPGD P15428 1/20 0.46
HTT P42858 1/20 0.46
PTGER1 P34995 2/20 0.45
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
CYP3A4 P08684 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2D6 P10635 1/20 0.43
OPRK1 P41145 1/20 0.43
BLM P54132 1/20 0.43
PMP22 Q01453 1/20 0.43
MAPT P10636 2/20 0.42
SMPD1 P17405 1/20 0.42
GAA P10253 1/20 0.41
PKM P14618 1/20 0.41
P4HB P07237 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8828260 0.91 OPRM1 (0.47) OPRM1TMEM97SIGMAR1LMNAHPGD
SCHEMBL8828362 0.89 LMNA (0.59) OPRM1TMEM97SIGMAR1LMNAHPGD
SCHEMBL8828302 0.88 LMNA (0.58) LMNAHPGDHTTKDM4EALDH1A1
SCHEMBL8828131 0.88 CYP3A4 (0.52) OPRM1TMEM97SIGMAR1HPGDKDM4E
SCHEMBL8828550 0.87 OPRM1 (0.49) OPRM1TMEM97SIGMAR1LMNAHPGD
SCHEMBL9047487 0.84 MEN1 (0.51) OPRM1TMEM97SIGMAR1LMNAHPGD
SCHEMBL8828184 0.84 OPRM1 (0.49) OPRM1TMEM97SIGMAR1HPGDKDM4E
SCHEMBL8828322 0.83 ALDH1A1 (0.56) OPRM1TMEM97SIGMAR1LMNAHPGD
SCHEMBL8828147 0.83 MAPT (0.56) OPRM1TMEM97SIGMAR1LMNAHPGD
SCHEMBL8828235 0.83 MAPT (0.56) OPRM1TMEM97SIGMAR1LMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5607953-A ANTIISCHEMIC AGENTS EISAI CO., LTD. (JP) 1997-03-04 US disclosed
EP-0344577-B1 Butenoic or propenoic acid derivatives EISAI CO LTD (JP) 1996-10-09 EP disclosed
US-5382595-A Antiischemic agents EISAI CO., LTD. (JP) 1995-01-17 US disclosed
US-5177089-A Antiischemic agent, vasodilator EISAI CO., LTD. (JP) 1993-01-05 US disclosed
EP-0344577-A2 Butenoic or propenoic acid derivatives Eisai Co., Ltd. (JP) 1989-12-06 EP disclosed