SCHEMBL8842827

SCHEMBL8842827

O=C(O)c1[nH]nc(-c2ccc(Cl)c(C(F)(F)F)c2)c1O

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 9/20 0.48
CYP1A2 P05177 1/20 0.48
KDR P35968 2/20 0.42
KDM2B Q8NHM5 1/20 0.42
KDM4C Q9H3R0 1/20 0.42
RORB Q92753 1/20 0.42
COMT P21964 1/20 0.41
HSP90AA1 P07900 1/20 0.41
PDE3B Q13370 1/20 0.40
PDE3A Q14432 1/20 0.40
SLC22A12 Q96S37 1/20 0.40
GYS1 P13807 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8842830 0.83 KIF11 (0.47)
SCHEMBL8842891 0.76 PIN1 (0.47) NOTUM
SCHEMBL8842823 0.71 RAB9A (0.50) CYP1A2
SCHEMBL2698021 0.68 NOTUM (0.61) NOTUMCYP1A2KDRCOMTPDE3B
SCHEMBL18955875 0.67 MAPT (0.42) NOTUMCYP1A2KDRKDM2BKDM4C
SCHEMBL375961 0.66 TSHR (0.59) NOTUMKDRKDM2BKDM4C
SCHEMBL322688 0.66 KIF11 (0.59) NOTUMCYP1A2KDRCOMT
SCHEMBL27355471 0.66 NOTUM (0.49) NOTUMCYP1A2KDM2BKDM4CRORB
SCHEMBL11622285 0.66 KDR (0.68) NOTUMCYP1A2KDRPDE3BPDE3A
SCHEMBL15012259 0.66 NOTUM (0.50) NOTUMCYP1A2RORBCOMTPDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5674887-A Prevention of bone resorption ELI LILLY AND COMPANY (US) 1997-10-07 US disclosed
EP-0578477-B1 Treatment of inflammatory bowel disease LILLY CO ELI (US) 1996-06-19 EP disclosed
US-5436258-A Prevention of bone resorption ELI LILLY AND COMPANY (US) 1995-07-25 US disclosed
EP-0587378-A1 Prevention of bone resorption ELI LILLY AND COMPANY (US) 1994-03-16 EP disclosed
US-5294630-A Treatment of inflammatory bowel disease ELI LILLY AND COMPANY (US) 1994-03-15 US disclosed
EP-0578477-A1 Treatment of inflammatory bowel disease ELI LILLY AND COMPANY (US) 1994-01-12 EP disclosed