SCHEMBL8863993

SCHEMBL8863993

CC(c1ccccc1Br)[N+](=O)[O-]

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.40
TP53 P04637 1/20 0.37
GAA P10253 1/20 0.37
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA9 Q16790 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C19 P33261 2/20 0.35
CYP2C9 P11712 1/20 0.35
HSD11B1 P28845 1/20 0.35
IDO1 P14902 1/20 0.34
TDO2 P48775 1/20 0.34
ALDH1A1 P00352 5/20 0.34
MAPT P10636 2/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CYP3A4 P08684 1/20 0.33
ALOX15 P16050 1/20 0.33
CTSB P07858 1/20 0.33
HSD17B10 Q99714 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27937647 0.78 HTT (0.43) HTTTP53GAACA1CA2
SCHEMBL7732490 0.78 CYP1A2 (0.40) HTTTP53GAACYP1A2CYP2C19
SCHEMBL5623819 0.78 ADRB2 (0.41) GAACYP1A2CYP2C19CYP2C9IDO1
SCHEMBL27496185 0.76 ALDH1A1 (0.53) CYP1A2ALDH1A1MAPTSMN1; SMN2HSD17B10
SCHEMBL10898417 0.76 GABRA1 (0.54) GAACA12CA1CA2CA9
SCHEMBL943534 0.74 MAPT (0.40) CA12CA1CA2CA9CYP1A2
SCHEMBL6029216 0.74 L3MBTL1 (0.43) GAACA1CA2ALDH1A1MAPT
SCHEMBL265334 0.74 ALDH1A1 (0.50) GAACYP1A2CYP2C19CYP2C9ALDH1A1
SCHEMBL11523492 0.73 CYP1A2 (0.39) CA1CA2CYP1A2ALDH1A1CYP3A4
SCHEMBL1044900 0.73 HTT (0.47) HTTGAACA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5691323-A BENZIMIDAZOL-2-ONES MERCK & CO., INC. (US) 1997-11-25 US disclosed
US-5574044-A BENZIMIDAZOL-2-ONE COMPOUNDS FOR TREATMENT OF MYOPIA MERCK & CO., INC. (US) 1996-11-12 US disclosed
WO-1996013262-A1 MUSCARINE ANTAGONISTS MERCK & CO., INC. (US) 1996-05-09 WO disclosed