SCHEMBL8879634

SCHEMBL8879634

CCOC(=O)c1nccn1C1Cc2c(F)cccc2C1=O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.37
SMN1; SMN2 Q16637 2/20 0.36
JAK2 O60674 1/20 0.36
JAK3 P52333 1/20 0.36
HPGD P15428 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
HSD17B10 Q99714 1/20 0.36
ADORA3 P0DMS8 1/20 0.35
ADORA2B P29275 1/20 0.35
GABRA1 P14867 2/20 0.35
GABRG2 P18507 2/20 0.35
GABRB3 P28472 2/20 0.35
GABRA5 P31644 2/20 0.35
GABRA3 P34903 2/20 0.35
MAPT P10636 2/20 0.34
MAPK1 P28482 1/20 0.34
ATM Q13315 1/20 0.34
KDM4E B2RXH2 2/20 0.34
GABRP O00591 1/20 0.34
GABRD O14764 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8881566 0.90 ACHE (0.40) ALDH1A1SMN1; SMN2HSD17B10ADORA3ADORA2B
SCHEMBL8880275 0.88 ADORA3 (0.35) SMN1; SMN2NPSR1ADORA3ADORA2BGABRA1
SCHEMBL8880778 0.88 MAPT (0.37) ALDH1A1SMN1; SMN2HPGDNPSR1ADORA3
SCHEMBL8883880 0.87 RAB9A (0.39) ALDH1A1SMN1; SMN2HPGDHSD17B10ADORA3
SCHEMBL8098958 0.86 ELANE (0.36) ALDH1A1HPGDHSD17B10ADORA3ADORA2B
SCHEMBL8012794 0.84 ELANE (0.34) ALDH1A1SMN1; SMN2ADORA3ADORA2BGABRA1
SCHEMBL8317836 0.84 TSHR (0.36) ALDH1A1SMN1; SMN2HPGDNPSR1HSD17B10
SCHEMBL8555959 0.84 KIF11 (0.34) POLB
SCHEMBL8879965 0.83 MAPT (0.46) ALDH1A1SMN1; SMN2HPGDHSD17B10ADORA3
SCHEMBL8556161 0.83 AADAT (0.34) MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5677306-A ANTAGONIZING ALPHA-AMINO-3-HYDROXY-5-METHYL-4-ISOXAZOLEPROPIONIC ACID RECEPTOR, USEFUL FOR TREATING ALL ISCHEMIAS RHONE-POULENC RORER S.A. (FR) 1997-10-14 US disclosed