SCHEMBL8897726

SCHEMBL8897726

O=c1ccc(-c2c(-c3cccc(-c4cccc(C(F)(F)F)c4)c3)n[nH]c2-c2ccccc2)n[nH]1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 1/20 0.46
NTRK1 P04629 1/20 0.46
RET P07949 1/20 0.46
PDGFRB P09619 1/20 0.46
CDK8 P49336 1/20 0.46
NTRK3 Q16288 1/20 0.46
NTRK2 Q16620 1/20 0.46
AURKB Q96GD4 1/20 0.46
MAPK14 Q16539 3/20 0.45
MAPK11 Q15759 2/20 0.45
MAPK13 O15264 1/20 0.45
RAF1 P04049 1/20 0.45
MAPK9 P45984 1/20 0.45
MAPK12 P53778 1/20 0.45
CYP1A2 P05177 1/20 0.45
PIM1 P11309 2/20 0.44
MAP4K4 O95819 1/20 0.44
GPX4 P36969 1/20 0.44
GSK3B P49841 1/20 0.44
PIM3 Q86V86 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8887885 0.82 CYP1A2 (0.50) MAPK14MAPK11MAPK13RAF1MAPK12
SCHEMBL8888361 0.80 CYP1A2 (0.50) PDGFRBCDK8NTRK3NTRK2AURKB
SCHEMBL8890194 0.80 CYP1A2 (0.50) MAPK14MAPK11MAPK13RAF1MAPK12
SCHEMBL8887621 0.80 CYP1A2 (0.50) MAPK14CYP1A2TP53MAPTSMN1; SMN2
SCHEMBL1769732 0.79 JAK2 (0.62) JAK2NTRK1RETPDGFRBCDK8
SCHEMBL8889484 0.77 CYP1A2 (0.53) MAPK14MAPK11MAPK13RAF1MAPK12
SCHEMBL8889663 0.77 CYP1A2 (0.47) CYP1A2TP53MAPTSMN1; SMN2AKR1B1
SCHEMBL8886941 0.77 NR1H2 (0.49) MAPK14MAPK11MAPK13RAF1MAPK12
SCHEMBL8889786 0.75 CYP1A2 (0.45) PDGFRBCDK8NTRK3NTRK2AURKB
SCHEMBL8888926 0.75 KMT2A (0.57) CYP1A2TP53MAPTSMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997001551-A1 PYRAZOLE COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-01-16 WO disclosed