SCHEMBL8890432

SCHEMBL8890432

Cn1c(=O)cc(N)n(-c2c(Cl)cc(C(F)(F)F)cc2Cl)c1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA2 P47869 17/20 0.43
GABRB2 P47870 17/20 0.43
GABRB3 P28472 17/20 0.43
GABRP O00591 16/20 0.43
GABRD O14764 16/20 0.43
GABRA1 P14867 16/20 0.43
GABRB1 P18505 16/20 0.43
GABRG2 P18507 16/20 0.43
GABRA5 P31644 16/20 0.43
GABRA3 P34903 16/20 0.43
GABRA4 P48169 16/20 0.43
GABRE P78334 16/20 0.43
GABRA6 Q16445 16/20 0.43
GABRG1 Q8N1C3 16/20 0.43
GABRG3 Q99928 16/20 0.43
GABRQ Q9UN88 16/20 0.43
CYP3A4 P08684 2/20 0.38
ALDH1A1 P00352 1/20 0.37
NR1I2 O75469 1/20 0.37
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29837238 0.70 GABRP (0.36) GABRA2GABRB2GABRB3GABRPGABRD
SCHEMBL26088331 0.70 GABRP (0.36) GABRA2GABRB2GABRB3GABRPGABRD
SCHEMBL8830715 0.69 CYP3A4 (0.50) CYP3A4ALDH1A1SMN1; SMN2
SCHEMBL9723057 0.69 ALDH1A1 (0.53) GABRA2GABRB2GABRB3GABRPGABRD
SCHEMBL10679118 0.68 GABRA2 (0.43) GABRA2GABRB2GABRB3GABRPGABRD
SCHEMBL10678078 0.68 GABRA2 (0.40) GABRA2GABRB2GABRB3GABRPGABRD
SCHEMBL10679158 0.68 GABRA2 (0.38) GABRA2GABRB2GABRB3GABRPGABRD
SCHEMBL8830700 0.68 ALDH1A1 (0.51) CYP3A4ALDH1A1SMN1; SMN2
SCHEMBL5867300 0.68 TLR8 (0.43) CYP3A4ALDH1A1SMN1; SMN2
SCHEMBL7801737 0.68 GABRB3 (0.48) GABRA2GABRB2GABRB3GABRPGABRD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997010220-A1 URACIL DERIVATIVE BAYER AKTIENGESELLSCHAFT (DE) 1997-03-20 WO disclosed