SCHEMBL8890567

SCHEMBL8890567

O=C(O)Cn1c(=O)[nH]c(=O)c2ccc(Br)cc21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 3/20 0.47
HDAC8 Q9BY41 3/20 0.47
HDAC6 Q9UBN7 3/20 0.47
AKR1A1 P14550 1/20 0.43
AKR1B1 P15121 1/20 0.43
GPR17 Q13304 1/20 0.40
EGLN1 Q9GZT9 1/20 0.39
GRIN2D O15399 2/20 0.39
GRIN3B O60391 2/20 0.39
GRIA1 P42261 2/20 0.39
GRIA2 P42262 2/20 0.39
GRIA3 P42263 2/20 0.39
GRIA4 P48058 2/20 0.39
GRIN1 Q05586 2/20 0.39
GRIN2A Q12879 2/20 0.39
GRIN2B Q13224 2/20 0.39
GRIN2C Q14957 2/20 0.39
GRIN3A Q8TCU5 2/20 0.39
GLA P06280 1/20 0.39
APEX1 P27695 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8046411 0.83 MAT2A (0.52) HDAC1HDAC8HDAC6AKR1A1AKR1B1
SCHEMBL4629626 0.82 B3GNT2 (0.47) GRIN2DGRIN3BGRIA1GRIA2GRIA3
SCHEMBL18554543 0.79 PDE5A (0.46) HDAC1HDAC8HDAC6AKR1A1AKR1B1
SCHEMBL8377270 0.79 KDM4E (0.64) AKR1B1GLAAPEX1KDM4E
SCHEMBL6358211 0.74 CBX7 (0.44) AKR1A1AKR1B1
SCHEMBL21027239 0.74 GLA (0.74) GLAAPEX1KDM4E
SCHEMBL21027247 0.73 GLA (0.51) AKR1A1AKR1B1EGLN1GLAKDM4E
SCHEMBL14692230 0.72 METAP2 (0.44) HDAC1HDAC8HDAC6EGLN1
SCHEMBL30015488 0.72 METAP2 (0.44) HDAC1HDAC8HDAC6EGLN1
SCHEMBL411220 0.72 KDM4E (0.56) AKR1A1AKR1B1GLAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997002254-A1 QUINAZOLINE DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-01-23 WO disclosed