SCHEMBL8891364

SCHEMBL8891364

OC(CNc1ccc2ccccc2c1)CN1CCN(c2cc(N3CCCC3)nc(N3CCCC3)n2)CC1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 13/20 0.49
CASP5 P51878 13/20 0.49
CASP4 P49662 11/20 0.47
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
TSHR P16473 1/20 0.41
GALR2 O43603 1/20 0.40
GALR1 P47211 1/20 0.40
MAPT P10636 1/20 0.39
KDM4E B2RXH2 1/20 0.39
USP2 O75604 1/20 0.39
MAPK1 P28482 1/20 0.39
HTT P42858 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
HSD17B10 Q99714 1/20 0.39
CNR1 P21554 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8891784 0.93 HRH4 (0.45) CASP1CASP5CASP4ALDH1A1LMNA
SCHEMBL8912652 0.81 CASP1 (0.58) CASP1CASP5CASP4ALDH1A1LMNA
SCHEMBL8892044 0.80 CASP1 (0.50) CASP1CASP5CASP4MAPT
SCHEMBL7769859 0.78 MAPT (0.60) TSHRMAPTKDM4EUSP2MAPK1
SCHEMBL8893240 0.76 RAD52 (0.46) ALDH1A1LMNAMAPTKDM4EMAPK1
SCHEMBL8890641 0.70 ABCB1 (0.50) ALDH1A1LMNAMAPTKDM4EMAPK1
SCHEMBL31536981 0.69 USP2 (0.46) LMNAMAPTKDM4EUSP2MAPK1
SCHEMBL31536985 0.69 DRD2 (0.48) USP2
SCHEMBL8890384 0.67 CASP1 (0.54) CASP1CASP5CASP4MAPT
SCHEMBL9129799 0.67 CASP1 (0.62) CASP1CASP5CASP4KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997014685-A1 PYRIMIDINE DERIVATIVES GYÓGYSZERKUTATÓ INTÉZET KFT (HU) 1997-04-24 WO disclosed