SCHEMBL8891784

SCHEMBL8891784

Nc1cc(N2CCN(CC(O)CNc3ccc4ccccc4c3)CC2)nc(N2CCCC2)n1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 2/20 0.45
CASP1 P29466 10/20 0.43
CASP5 P51878 10/20 0.43
CASP4 P49662 9/20 0.41
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
TSHR P16473 1/20 0.39
GALR2 O43603 1/20 0.38
GALR1 P47211 1/20 0.38
MAPT P10636 1/20 0.37
KDM4E B2RXH2 1/20 0.36
USP2 O75604 1/20 0.36
MAPK1 P28482 1/20 0.36
HTT P42858 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
HSD17B10 Q99714 1/20 0.36
CNR1 P21554 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8891364 0.93 CASP1 (0.49) CASP1CASP5CASP4ALDH1A1LMNA
SCHEMBL8912652 0.75 CASP1 (0.58) CASP1CASP5CASP4ALDH1A1LMNA
SCHEMBL8892044 0.74 CASP1 (0.50) CASP1CASP5CASP4MAPT
SCHEMBL7769859 0.73 MAPT (0.60) TSHRMAPTKDM4EUSP2MAPK1
SCHEMBL8893240 0.73 RAD52 (0.46) ALDH1A1LMNAMAPTKDM4EMAPK1
SCHEMBL10143607 0.69 HRH4 (0.81) HRH4CASP1CASP5CASP4LMNA
SCHEMBL4845325 0.68 KDM1A (0.47) ALDH1A1TSHRMAPTKDM4E
SCHEMBL10377525 0.67 HRH4 (0.78) HRH4CASP1CASP5CASP4LMNA
SCHEMBL8890641 0.67 ABCB1 (0.50) ALDH1A1LMNAMAPTKDM4EMAPK1
SCHEMBL10848170 0.66 CASP1 (0.75) HRH4CASP1CASP5CASP4LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997014685-A1 PYRIMIDINE DERIVATIVES GYÓGYSZERKUTATÓ INTÉZET KFT (HU) 1997-04-24 WO disclosed