SCHEMBL8891690

SCHEMBL8891690

CNC(=O)NS(=O)(=O)c1cc(CC(=O)NC(C)c2ccoc2)ccc1C

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.37
ALDH1A1 P00352 4/20 0.36
MAPT P10636 1/20 0.36
HPGD P15428 1/20 0.36
CA2 P00918 1/20 0.36
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
IDH1 O75874 2/20 0.34
CNR1 P21554 1/20 0.34
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8892002 0.90 HTT (0.36) HTTALDH1A1MAPTHPGDCA2
SCHEMBL8891613 0.89 KEAP1 (0.33) HTTALDH1A1MAPTCA2IDH1
SCHEMBL8891142 0.88 HTT (0.35) HTTALDH1A1MAPTHPGDCA2
SCHEMBL8893753 0.88 POLB (0.41) HTTALDH1A1CNR1MEN1KMT2A
SCHEMBL8891432 0.86 ALDH1A1 (0.37) HTTALDH1A1CNR1KMT2A
SCHEMBL8892270 0.85 KEAP1 (0.39) HTTALDH1A1MAPTHPGDMEN1
SCHEMBL8891731 0.83 HTT (0.38) HTTALDH1A1MAPTHPGDCA2
SCHEMBL8892494 0.83 HTT (0.38) HTTALDH1A1MAPTHPGDCA2
SCHEMBL8891913 0.83 KDM4E (0.43) HTTALDH1A1MAPTHPGDCA2
SCHEMBL8892189 0.80 LMNA (0.35) HTTALDH1A1MAPTHPGDCA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5607976-A ANNTIISCHEMIC AGENTS AND CARDIOVASCULAR DISORDERS HOECHST AKTIENGESELLSCHAFT (DE) 1997-03-04 US disclosed