SCHEMBL8893666

SCHEMBL8893666

CNC(=O)NS(=O)(=O)c1cc(CC(=O)NC(C)c2ccco2)ccc1SC

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.35
OPRM1 P35372 1/20 0.35
OPRD1 P41143 1/20 0.35
TP53 P04637 1/20 0.33
CA2 P00918 1/20 0.33
ALDH1A1 P00352 3/20 0.33
MAPT P10636 2/20 0.33
HPGD P15428 1/20 0.33
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
CCR2 P41597 1/20 0.32
HTT P42858 1/20 0.32
HSD17B10 Q99714 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
EGFR P00533 1/20 0.31
ERBB2 P04626 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8891256 0.91 KDM4E (0.34) KDM4EOPRM1OPRD1TP53CA2
SCHEMBL8891767 0.89 KDM4E (0.34) KDM4EOPRM1OPRD1TP53ALDH1A1
SCHEMBL8891913 0.87 KDM4E (0.43) KDM4EOPRM1OPRD1TP53CA2
SCHEMBL8898777 0.85 ALDH1A1 (0.41) KDM4EALDH1A1MAPTHPGDHSD17B10
SCHEMBL8891142 0.84 HTT (0.35) KDM4ECA2ALDH1A1MAPTHPGD
SCHEMBL8891063 0.83 LMNA (0.43) KDM4EALDH1A1MAPTHPGDHSD17B10
SCHEMBL8892045 0.82 CA2 (0.32) CA2ALDH1A1MAPTHPGDCYP3A4
SCHEMBL8890064 0.82 L3MBTL1 (0.43) TP53CA2ALDH1A1MAPTHPGD
SCHEMBL8892224 0.82 NPSR1 (0.45) KDM4EOPRM1OPRD1TP53ALDH1A1
SCHEMBL8893667 0.81 CCR2 (0.32) KDM4EOPRM1OPRD1CA2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5607976-A ANNTIISCHEMIC AGENTS AND CARDIOVASCULAR DISORDERS HOECHST AKTIENGESELLSCHAFT (DE) 1997-03-04 US disclosed