SCHEMBL8908590

SCHEMBL8908590

CCN(CC)CCSC1c2ccccc2-c2[nH]c(=O)c(=O)[nH]c21

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.36
ALDH1A1 P00352 7/20 0.35
HPGD P15428 4/20 0.35
ALOX12 P18054 1/20 0.35
MAPT P10636 2/20 0.33
KMT2A Q03164 2/20 0.32
MEN1 O00255 1/20 0.32
CHRM2 P08172 1/20 0.32
CHRM4 P08173 1/20 0.32
CHRM1 P11229 1/20 0.32
CHRM3 P20309 1/20 0.32
KDM4E B2RXH2 5/20 0.32
POLB P06746 2/20 0.31
ALOX15 P16050 1/20 0.31
NPC1 O15118 2/20 0.31
MITF O75030 2/20 0.31
RAB9A P51151 2/20 0.31
DNMT1 P26358 1/20 0.31
HTT P42858 1/20 0.31
RAD52 P43351 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8907599 0.67 CYP1A2 (0.38) TSHRALDH1A1MAPTKDM4EPOLB
SCHEMBL8907689 0.65 SERPINE1 (0.36) ALDH1A1MAPTKMT2AMEN1KDM4E
SCHEMBL8907884 0.65 S100A4 (0.36) TSHRALDH1A1HPGDKDM4EPOLB
SCHEMBL8909107 0.62 TSHR (0.33) TSHRALDH1A1HPGDALOX12MAPT
SCHEMBL8908307 0.61 ACP3 (0.40) ALDH1A1KDM4EPOLBRAB9AAPAF1
SCHEMBL1107119 0.61 ACHE (0.47) ALDH1A1MAPTKMT2AMEN1CHRM2
SCHEMBL10880774 0.60 TBXA2R (0.40)
SCHEMBL2763720 0.59 SERPINE1 (0.35) ALDH1A1HPGDKMT2AMEN1KDM4E
SCHEMBL8908407 0.59 ALDH1A1 (0.39) TSHRALDH1A1POLBSMN1; SMN2
SCHEMBL11647247 0.57 PARP3 (0.42) ALDH1A1HPGDALOX12KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0682657-B1 9H-INDENO[1,2-b]PYRAZINE-3(4H)-ONES AND 9H-INDENO[1,2-b]PYRAZINE-2,3(1H,4H)-DIONES AND THEIR PREPARATION AND USE NOVO NORDISK AS (DK) 1997-11-19 EP claimed
US-5646146-A CENTRAL NERVOUS SYSTEM DISORDERS NOVO NORDISK A/S (DK) 1997-07-08 US claimed