SCHEMBL8908933

SCHEMBL8908933

O=c1[nH]c2c([nH]c1=O)C(N1CCNCC1)c1ccccc1-2

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 5/20 0.40
HTR2B P41595 5/20 0.40
HTR2A P28223 4/20 0.40
GAA P10253 2/20 0.36
USP2 O75604 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
TSHR P16473 1/20 0.36
CYP2C19 P33261 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CACNA1G O43497 1/20 0.35
TAAR1 Q96RJ0 1/20 0.35
ALDH1A1 P00352 1/20 0.34
POLB P06746 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
LMNA P02545 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8908407 0.85 ALDH1A1 (0.39) HTR2CHTR2BHTR2AGAAUSP2
SCHEMBL8908855 0.85 CYP1A2 (0.44) GAAUSP2CYP1A2CYP3A4CYP2D6
SCHEMBL8908279 0.80 RAB9A (0.46) HTR2CHTR2BHTR2AGAACYP2D6
SCHEMBL8908448 0.80 ALDH1A1 (0.43) GAAUSP2CYP1A2CYP3A4CYP2D6
SCHEMBL1798685 0.77 CYP1A2 (0.53) HTR2CHTR2BHTR2AGAACYP1A2
SCHEMBL8909181 0.76 HTR2C (0.49) HTR2CHTR2ACYP3A4CYP2D6CYP2C19
Hydrochloric Acid SCHEMBL6167962 0.75 CYP1A2 (0.52) HTR2CHTR2BHTR2AGAACYP1A2
SCHEMBL6992174 0.70 CYP1A2 (0.46) HTR2CHTR2BHTR2AUSP2CYP1A2
SCHEMBL8907689 0.69 SERPINE1 (0.36) HTR2BCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL8907884 0.69 S100A4 (0.36) TSHRSMN1; SMN2ALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0682657-B1 9H-INDENO[1,2-b]PYRAZINE-3(4H)-ONES AND 9H-INDENO[1,2-b]PYRAZINE-2,3(1H,4H)-DIONES AND THEIR PREPARATION AND USE NOVO NORDISK AS (DK) 1997-11-19 EP disclosed