SCHEMBL8912282

SCHEMBL8912282

Cc1nc(N)[nH]c(=O)c1N1CCN(c2ccccc2C#N)CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 5/20 0.43
DRD2 P14416 4/20 0.42
DRD3 P35462 2/20 0.42
AR P10275 1/20 0.41
HTR1A P08908 3/20 0.40
ADRA1A P35348 2/20 0.40
ADRA1B P35368 2/20 0.40
HTR7 P34969 2/20 0.40
ADRA1D P25100 1/20 0.40
PHGDH O43175 1/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
HTR2A P28223 1/20 0.40
THPO P40225 1/20 0.40
HIF1A Q16665 1/20 0.40
GRM5 P41594 1/20 0.40
DHFR P00374 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8911693 0.81 TTR (0.47) ALDH1A1CYP1A2HIF1ADHFRXDH
SCHEMBL8912815 0.75 TSHR (0.57) DRD4DRD2DRD3KDM4EALDH1A1
SCHEMBL8912435 0.71 DHFR (0.40) DHFRXDHNOS1
SCHEMBL8913183 0.71 DHFR (0.44) DHFRXDHNOS1
SCHEMBL3088832 0.71 DRD4 (0.54) DRD4DRD2DRD3ARHTR1A
SCHEMBL8912802 0.69 SIRT6 (0.50) ALDH1A1DHFR
SCHEMBL20139817 0.68 RXFP1 (0.52) DRD4DRD2DRD3ARPHGDH
SCHEMBL20140652 0.68 PHGDH (0.45) DRD4DRD2DRD3ARHTR1A
SCHEMBL6261764 0.68 DRD4 (0.45) DRD4DRD2DRD3ARKDM4E
SCHEMBL20139913 0.67 DRD4 (0.47) DRD4DRD2DRD3ARHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5670508-A ANTITUMOR AGENTS FOR BRAIN TUMORS NATIONAL SCIENCE COUNCIL (TW) 1997-09-23 US disclosed