SCHEMBL8922784

SCHEMBL8922784

O=C(O)c1c(N2CCOCC2)c(-c2ccccc2)cn1Cc1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.45
ALDH1A1 P00352 7/20 0.44
HPGD P15428 2/20 0.44
ALOX15 P16050 1/20 0.44
PKM P14618 2/20 0.43
RAB9A P51151 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
SMN1; SMN2 Q16637 3/20 0.41
NPC1 O15118 1/20 0.41
PIK3CD O00329 1/20 0.41
PIK3CA P42336 1/20 0.41
PIK3CB P42338 1/20 0.41
PIK3CG P48736 1/20 0.41
MAPT P10636 2/20 0.40
KDM4E B2RXH2 1/20 0.40
LMNA P02545 1/20 0.40
HTT P42858 1/20 0.40
PDE10A Q9Y233 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
CYP1A2 P05177 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8922826 0.93 ALDH1A1 (0.43) HSD17B10ALDH1A1HPGDALOX15PKM
SCHEMBL9857292 0.82 ALDH1A1 (0.44) HSD17B10ALDH1A1HPGDALOX15PKM
SCHEMBL8925211 0.80 ALDH1A1 (0.54) HSD17B10ALDH1A1HPGDALOX15SMN1; SMN2
SCHEMBL8922256 0.80 HSD17B10 (0.49) HSD17B10ALDH1A1HPGDALOX15TDP1
SCHEMBL8923374 0.76 ALDH1A1 (0.40) HSD17B10ALDH1A1HPGDALOX15RAB9A
SCHEMBL8923602 0.72 PIK3CA (0.42) ALDH1A1RAB9ATDP1SMN1; SMN2NPC1
SCHEMBL8922352 0.70 ALDH1A1 (0.41) HSD17B10ALDH1A1HPGDALOX15PKM
SCHEMBL8920356 0.69 AKR1C3 (0.40) HSD17B10ALDH1A1HPGDALOX15RAB9A
SCHEMBL8920563 0.68 ALDH1A1 (0.70) HSD17B10ALDH1A1HPGDALOX15SMN1; SMN2
SCHEMBL9857777 0.67 ALDH1A1 (0.47) HSD17B10ALDH1A1HPGDALOX15RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5684160-A 3-aminopyrroles, methods for their synthesis and for their pharmaceutical use ARZNEIMETTELWERK DRESDEN GMBH (DE) 1997-11-04 US claimed
US-5502051-A CENTRAL NERVOUS SYSTEM, ANTISPASMODIC ARZNEIMITTELWERK DRESDEN GMBH (DE) 1996-03-26 US claimed
EP-0431371-A1 3-Aminopyrroles, process for this preparation and their use as medicaments ARZNEIMITTELWERK DRESDEN GmbH (DE) 1991-06-12 EP claimed
US-5684160-A 3-aminopyrroles, methods for their synthesis and for their pharmaceutical use ARZNEIMETTELWERK DRESDEN GMBH (DE) 1997-11-04 US disclosed
US-5502051-A CENTRAL NERVOUS SYSTEM, ANTISPASMODIC ARZNEIMITTELWERK DRESDEN GMBH (DE) 1996-03-26 US disclosed