SCHEMBL8922352

SCHEMBL8922352

Cc1ccc(-c2cn(C)c(C(=O)O)c2N2CCOCC2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.41
HPGD P15428 3/20 0.41
USP2 O75604 1/20 0.41
FKBP1A P62942 1/20 0.41
CHRNA7 P36544 1/20 0.41
AKR1C3 P42330 1/20 0.41
CYP2D6 P10635 1/20 0.41
HSD17B10 Q99714 2/20 0.41
ALOX15 P16050 1/20 0.41
PIK3CA P42336 2/20 0.40
PIK3CG P48736 2/20 0.40
MTOR P42345 1/20 0.40
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
ATM Q13315 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
TP53 P04637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8922256 0.90 HSD17B10 (0.49) ALDH1A1HPGDUSP2CHRNA7CYP2D6
SCHEMBL8920356 0.89 AKR1C3 (0.40) ALDH1A1HPGDAKR1C3HSD17B10ALOX15
SCHEMBL8923602 0.89 PIK3CA (0.42) ALDH1A1AKR1C3PIK3CAPIK3CGMTOR
SCHEMBL9857290 0.81 POLB (0.43) ALDH1A1HPGDUSP2FKBP1ACHRNA7
SCHEMBL8923375 0.74 ALDH1A1 (0.63) ALDH1A1HPGDUSP2FKBP1ACHRNA7
SCHEMBL8923374 0.73 ALDH1A1 (0.40) ALDH1A1HPGDAKR1C3HSD17B10ALOX15
SCHEMBL9857777 0.71 ALDH1A1 (0.47) ALDH1A1HPGDUSP2CHRNA7HSD17B10
SCHEMBL8925211 0.70 ALDH1A1 (0.54) ALDH1A1HPGDHSD17B10ALOX15KDM4E
SCHEMBL8922784 0.70 HSD17B10 (0.45) ALDH1A1HPGDFKBP1AHSD17B10ALOX15
SCHEMBL8922826 0.69 ALDH1A1 (0.43) ALDH1A1HPGDAKR1C3HSD17B10ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5684160-A 3-aminopyrroles, methods for their synthesis and for their pharmaceutical use ARZNEIMETTELWERK DRESDEN GMBH (DE) 1997-11-04 US claimed
US-5502051-A CENTRAL NERVOUS SYSTEM, ANTISPASMODIC ARZNEIMITTELWERK DRESDEN GMBH (DE) 1996-03-26 US claimed
EP-0431371-A1 3-Aminopyrroles, process for this preparation and their use as medicaments ARZNEIMITTELWERK DRESDEN GmbH (DE) 1991-06-12 EP claimed
US-5684160-A 3-aminopyrroles, methods for their synthesis and for their pharmaceutical use ARZNEIMETTELWERK DRESDEN GMBH (DE) 1997-11-04 US disclosed
US-5502051-A CENTRAL NERVOUS SYSTEM, ANTISPASMODIC ARZNEIMITTELWERK DRESDEN GMBH (DE) 1996-03-26 US disclosed