SCHEMBL8933547

SCHEMBL8933547

CC(=O)c1ccc2c(c1)C(c1ccccc1F)=NCC(NCC1(CO)OCCO1)=N2

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNE2 O96020 1/20 0.34
CCNE1 P24864 1/20 0.34
CDK2 P24941 1/20 0.34
ALDH1A1 P00352 3/20 0.32
MAPT P10636 3/20 0.32
NPC1 O15118 2/20 0.32
RAB9A P51151 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
GABRA1 P14867 2/20 0.32
GABRA5 P31644 2/20 0.32
GABRA3 P34903 2/20 0.32
GABRA2 P47869 2/20 0.32
GABRB2 P47870 2/20 0.32
MEN1 O00255 1/20 0.32
NFKB1 P19838 1/20 0.32
NFKB2 Q00653 1/20 0.32
KMT2A Q03164 1/20 0.32
RELA Q04206 1/20 0.32
LMNA P02545 1/20 0.32
CCKBR P32239 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8933416 0.79 GABRA3 (0.35) ALDH1A1MAPTNPC1RAB9ASMN1; SMN2
SCHEMBL8933545 0.76 CCNE2 (0.42) CCNE2CCNE1CDK2ALDH1A1MAPT
SCHEMBL11714852 0.74 OPRK1 (0.41) ALDH1A1MAPTSMN1; SMN2GABRA1GABRA5
SCHEMBL11454061 0.68 LMNA (0.48) LMNATP53AURKA
SCHEMBL8933492 0.67 GABRA1 (0.67) CCNE2CCNE1CDK2GABRA1GABRA5
SCHEMBL11830651 0.67 GABRA3 (0.42) CCNE2CCNE1CDK2GABRA1GABRA5
SCHEMBL8933535 0.67 CHRM1 (0.66) CCNE2CCNE1CDK2ALDH1A1SMN1; SMN2
SCHEMBL7348170 0.66 TP53 (0.38) ALDH1A1MAPTNPC1RAB9ASMN1; SMN2
SCHEMBL11749036 0.66 CYP3A4 (0.43) LMNAAURKA
SCHEMBL11445395 0.66 GABRA1 (0.50) ALDH1A1MAPTNPC1RAB9AGABRA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996023790-A1 ACETYLIMIDAZOBENZODIAZEPINES F. HOFFMANN-LA ROCHE AG (CH) 1996-08-08 WO disclosed