Fumaric Acid

Fumaric Acid

SCHEMBL8934540

Cc1ccn2c(C)c(CCc3cccc(NC4=NCCS4)c3)nc2c1.O=C(O)/C=C/C(=O)O.O=C(O)/C=C/C(=O)O

nearest known ligand 0.39

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADRB1ADRB2ATP4AATP4BAXLCHRM2CHRM3DRD2FLT3HRH1HTR2AHTR2BHTR2CKCNH2KMT2AMAP2K1MAP2K2MEN1MLNRPLK4RENS1PR1SLC6A2SLC6A4atpAatpBatpCatpDatpEatpFatpFHatpGpol

The experimentally established mechanism targets of Fumaric Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A known ✓ Q03164 2/20 0.33
MEN1 known ✓ O00255 1/20 0.32
MAPT P10636 3/20 0.39
MCL1 Q07820 2/20 0.39
TDP1 Q9NUW8 2/20 0.39
LMNA P02545 1/20 0.39
RECQL P46063 1/20 0.39
ATM Q13315 1/20 0.39
POLB P06746 2/20 0.37
TP53 P04637 2/20 0.37
RXFP1 Q9HBX9 1/20 0.37
NPC1 O15118 4/20 0.37
RAB9A P51151 4/20 0.37
KDM4E B2RXH2 1/20 0.37
AOC3 Q16853 1/20 0.36
NPY1R P25929 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.34
NFKB1 P19838 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fumaric Acid SCHEMBL8934542 1.00 MAPT (0.39) MAPTMCL1TDP1LMNARECQL
SCHEMBL8934533 0.82 NPY1R (0.50) POLBAOC3NPY1RSMN1; SMN2HPGD
SCHEMBL8934504 0.73 NPY1R (0.48) POLBAOC3NPY1RSMN1; SMN2HPGD
SCHEMBL8934581 0.68 TP53 (0.36) MAPTTDP1LMNAPOLBTP53
SCHEMBL8934543 0.68 MAOA (0.43) MAPTLMNAPOLBTP53RXFP1
SCHEMBL9628581 0.65 POLB (0.51) ATMPOLBNPY1RSMN1; SMN2KMT2A
SCHEMBL8934556 0.64 ADRA2A (0.48) AOC3
SCHEMBL8934518 0.64 NPY1R (0.50) TDP1LMNAPOLBKDM4EAOC3
SCHEMBL8934592 0.64 MAPT (0.37) MAPTTDP1POLBTP53RXFP1
SCHEMBL9378184 0.64 MAPT (0.41) MAPTPOLBTP53RXFP1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996030350-A1 AMIDINE DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-10-03 WO disclosed