SCHEMBL8941935

SCHEMBL8941935

COc1ccc(N2C(=O)O[C@H](COc3ccc(C=O)cc3)[C@@H]2C)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.44
CYP2A6 P11509 1/20 0.44
GRM2 Q14416 3/20 0.41
HSD11B1 P28845 3/20 0.36
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
USP2 O75604 2/20 0.36
TDP1 Q9NUW8 2/20 0.36
CLK1 P49759 1/20 0.36
DYRK1A Q13627 1/20 0.36
DYRK1B Q9Y463 1/20 0.36
MIF P14174 1/20 0.35
XDH P47989 1/20 0.34
TSHR P16473 2/20 0.34
MAPK1 P28482 2/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C19 P33261 1/20 0.34
MAPT P10636 3/20 0.34
HPGD P15428 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8941897 0.85 GRM2 (0.42) ALDH1A1GRM2HSD11B1MEN1KMT2A
SCHEMBL8941889 0.82 PIM1 (0.56) CLK1DYRK1ADYRK1BHPGDATM
SCHEMBL8941864 0.77 HSD11B1 (0.43) GRM2HSD11B1MEN1KMT2ASMN1; SMN2
SCHEMBL8941893 0.75 CSNK2A2 (0.48) GRM2MEN1KMT2ACLK1DYRK1A
SCHEMBL8942109 0.75 FFAR1 (0.50) ALDH1A1MEN1KMT2ATDP1TSHR
SCHEMBL8942112 0.72 SIRT2 (0.37) GRM2MAPTLMNA
SCHEMBL4467710 0.69 GRM2 (0.46) GRM2HSD11B1MEN1KMT2ATDP1
SCHEMBL8470701 0.68 ALDH1A1 (0.47) ALDH1A1CYP2A6GRM2MEN1KMT2A
SCHEMBL14996346 0.67 ALDH1A1 (0.76) ALDH1A1CYP2A6MEN1KMT2ATDP1
SCHEMBL19214413 0.67 ALDH1A1 (0.76) ALDH1A1CYP2A6TDP1MAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5521202-A ANTIDIABETIC AGENTS TAIHO PHARMACEUTICAL CO., LTD. (JP) 1996-05-28 US disclosed
EP-0645387-A1 THIAZOLIDINE DERIVATIVE AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME TAIHO PHARMACEUTICAL CO., LTD. (JP) 1995-03-29 EP disclosed