SCHEMBL8946339

SCHEMBL8946339

CCCCOC(=O)c1cc(NC)c2c(Cl)cc(Cl)cc2n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 2/20 0.42
KMT2A Q03164 2/20 0.38
MEN1 O00255 1/20 0.38
L3MBTL1 Q9Y468 4/20 0.38
TSHR P16473 3/20 0.38
TDP1 Q9NUW8 2/20 0.38
ALDH1A1 P00352 3/20 0.38
NQO2 P16083 2/20 0.38
LMNA P02545 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
KDM4E B2RXH2 2/20 0.36
POLB P06746 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
MAPT P10636 1/20 0.36
CYP2C9 P11712 1/20 0.36
HPGD P15428 1/20 0.36
CYP2C19 P33261 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CNR1 P21554 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8946246 0.88 CYP1A2 (0.42) TDP1ALDH1A1NQO2LMNACYP1A2
SCHEMBL8946290 0.83 NQO2 (0.53) ALDH1A1NQO2KDM4EPOLB
SCHEMBL8946957 0.82 NQO2 (0.39) KMT2AMEN1L3MBTL1TSHRALDH1A1
SCHEMBL8946276 0.78 ACHE (0.40) NQO2
SCHEMBL9380614 0.74 HTR3A (0.40) KMT2AMEN1TSHRNQO2LMNA
SCHEMBL9462723 0.72 NQO2 (0.52) ALDH1A1NQO2KDM4ECYP1A2HPGD
SCHEMBL1615754 0.71 ALDH1A1 (0.46) KMT2AMEN1ALDH1A1NQO2POLB
SCHEMBL29617388 0.71 ALDH1A1 (0.46) KMT2AMEN1ALDH1A1NQO2POLB
SCHEMBL1617936 0.70 GABRA2 (0.42) KMT2AMEN1L3MBTL1TDP1ALDH1A1
SCHEMBL17372709 0.70 MAPT (0.45) L3MBTL1ALDH1A1POLBMAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5493027-A ANTIEPILEPTIC AGENTS, NEUROGENATIVE DISEASES BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 1996-02-20 US disclosed