SCHEMBL8950221

SCHEMBL8950221

CCOC(=O)CN(c1cccc(OC)c1)S(=O)(=O)c1sccc1C1OCCO1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.45
LMNA P02545 6/20 0.40
ESR1 P03372 1/20 0.40
KMT2A Q03164 3/20 0.38
MAPT P10636 3/20 0.38
MEN1 O00255 2/20 0.38
ALDH1A1 P00352 5/20 0.37
NPSR1 Q6W5P4 1/20 0.37
MTNR1A P48039 1/20 0.36
MTNR1B P49286 1/20 0.36
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
ALOX15 P16050 1/20 0.35
CYP2C19 P33261 1/20 0.35
GAA P10253 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
TSHR P16473 1/20 0.35
MAPK1 P28482 1/20 0.35
USP2 O75604 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8950198 0.79 GAA (0.36) HTTKMT2AMAPTMEN1ALDH1A1
SCHEMBL8950073 0.79 ALDH1A1 (0.55) LMNAMAPTALDH1A1GAA
SCHEMBL8950311 0.77 ALDH1A1 (0.34) LMNAKMT2AMAPTMEN1ALDH1A1
SCHEMBL8862623 0.70 ALDH1A1 (0.43) ALDH1A1NPSR1CYP3A4CYP2C9CYP2C19
SCHEMBL8950605 0.69 LMNA (0.47) HTTLMNAKMT2AMAPTMEN1
SCHEMBL10011062 0.67 MTNR1A (0.55) LMNAMAPTALDH1A1MTNR1AMTNR1B
SCHEMBL8950386 0.65 GAA (0.38) HTTLMNAKMT2AMAPTMEN1
SCHEMBL7000752 0.65 KEAP1 (0.66) HTTLMNAKMT2AMAPTMEN1
SCHEMBL28970975 0.64 KDM4E (0.52) HTTLMNAMAPTALDH1A1MTNR1A
SCHEMBL7003143 0.63 KEAP1 (0.71) LMNAKMT2AMAPTMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996022099-A1 OPHTHALMIC COMPOSITIONS FOR TREATING GLAUCOMA ALCON LABORATORIES, INC. (US) 1996-07-25 WO disclosed
US-5538966-A ENZYME INHIBITORS FOR TREATMENT OF GLAUCOMA ALCON LABORATORIES, INC. (US) 1996-07-23 US disclosed
WO-1995019981-A1 THIENOTHIAZINE SULFONAMIDE DERIVATIVES PROCESS AND INTERMEDIATES FOR THEIR PREPARATION AND THEIR USE AS CARBONIC ANHYDRASE INHIBITORS ALCON LABORATORIES, INC. (US) 1995-07-27 WO disclosed