SCHEMBL8954337

SCHEMBL8954337

CCCCc1nc(Cc2ccccc2Cl)c(CC(Cc2ccccc2)C(=O)OC)[nH]1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.38
PARP1 P09874 2/20 0.37
APLNR P35414 1/20 0.37
PARP3 Q9Y6F1 1/20 0.37
POLB P06746 1/20 0.36
NOS3 P29474 1/20 0.35
NOS1 P29475 1/20 0.35
NOS2 P35228 1/20 0.35
ALOX5 P09917 2/20 0.35
BIRC2 Q13490 1/20 0.35
KMT2A Q03164 1/20 0.35
PTGES O14684 1/20 0.35
PYGL P06737 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
HPGD P15428 1/20 0.35
CYP2C19 P33261 1/20 0.35
HTT P42858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28161278 0.79 PARP1 (0.41) PARP1APLNRHTT
SCHEMBL9509544 0.78 APLNR (0.40) PARP1APLNRALOX5PTGESHTT
SCHEMBL9529092 0.77 PARP1 (0.35) PARP1
SCHEMBL9512926 0.76 HPGD (0.41) PARP1APLNRHPGDHTT
SCHEMBL9530397 0.75 BRS3 (0.40) ALOX5PTGESCYP1A2
Hydrochloric Acid SCHEMBL9267601 0.74 PARP1 (0.39) PARP1APLNRHPGDHTT
SCHEMBL9529061 0.72 CYP1A2 (0.39) PARP1ALOX5PTGESCYP1A2
SCHEMBL8954087 0.72
SCHEMBL8741912 0.69 AGTR1 (0.36) PARP1APLNR
SCHEMBL9052148 0.67 PARP1 (0.40) PARP1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5530017-A CONGESTIVE HEART FAILURE, RENAL FAILURE AND GLAUCOMA SMITHKLINE BEECHAM CORP (US) 1996-06-25 US disclosed
US-5444080-A Hypotensive agents SMITHKLINE BEECHAM CORPORATION (US) 1995-08-22 US disclosed
EP-0541705-A4 SUBSTITUTED 1H-IMIDAZOL-5-YL)ALKANOIC ACIDS 1993-11-10 EP disclosed
EP-0541705-A1 SUBSTITUTED 1H-IMIDAZOL-5-YL]ALKANOIC ACIDS SMITHKLINE BEECHAM CORPORATION (US) 1993-05-19 EP disclosed
WO-1992002510-A1 SUBSTITUTED [1H-IMIDAZOL-5-YL]ALKANOIC ACIDS SMITHKLINE BEECHAM CORPORATION (US) 1992-02-20 WO disclosed