SCHEMBL8957358

SCHEMBL8957358

NNC(=O)CCCCCCCCCCNC(=O)COc1ccc(CC(CN(CCN(CC(=O)O)CC(=O)O)CC(=O)O)N(CC(=O)O)CC(=O)O)cc1

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 1/20 0.45
ITGA2B P08514 1/20 0.45
EPOR P19235 2/20 0.38
FOLH1 Q04609 1/20 0.37
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CA1 P00915 6/20 0.35
CA2 P00918 6/20 0.35
CA12 O43570 2/20 0.35
CA9 Q16790 2/20 0.35
CYP3A4 P08684 1/20 0.35
KDM4E B2RXH2 1/20 0.35
TSHR P16473 1/20 0.35
RECQL P46063 1/20 0.35
PTPN1 P18031 1/20 0.35
CA4 P22748 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8957356 0.95 ITGB3 (0.47) ITGB3ITGA2BEPORFOLH1CYP1A2
SCHEMBL8842428 0.88 ALDH1A1 (0.41) CA1CA2CA12CA9KDM4E
SCHEMBL6047694 0.83 EPOR (0.40) ITGB3ITGA2BEPORFOLH1CA1
SCHEMBL6047708 0.83 EPOR (0.40) ITGB3ITGA2BEPORFOLH1CA1
SCHEMBL8842690 0.83 ALDH1A1 (0.40) CA1CA2CA12CA9KDM4E
SCHEMBL8842421 0.83 ALDH1A1 (0.43) KDM4E
SCHEMBL8957288 0.81 ITGB3 (0.44) ITGB3ITGA2BEPORCYP1A2CYP2D6
SCHEMBL8957385 0.81 ADRB1 (0.37) CYP1A2
SCHEMBL8092343 0.80 MAOB (0.41) TSHR
SCHEMBL8378153 0.78 LMNA (0.44) EPORFOLH1CA1CA2CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5482700-A Substituted polyamino, polycarboxy complexing agent dimers for MRI and X-ray contrast SCHERING AKTIENGESELLSCHAFT (DE) 1996-01-09 US disclosed
EP-0357622-A1 SUBSTITUTED COMPLEX-FORMING SUBSTANCES, COMPLEXES AND COMPLEX SALTS, PROCESS FOR MANUFACTURE THEREOF AND PHARMACEUTICAL AGENTS WHICH CONTAIN THEM SCHERING AKTIENGESELLSCHAFT (DE) 1990-03-14 EP disclosed
WO-1988007521-A1 SUBSTITUTED COMPLEX-FORMING SUBSTANCES, COMPLEXES AND COMPLEX SALTS, PROCESS FOR MANUFACTURE THEREOF AND PHARMACEUTICAL AGENTS WHICH CONTAIN THEM SCHERING AKTIENGESELLSCHAFT (DE) 1988-10-06 WO disclosed