SCHEMBL8968376

SCHEMBL8968376

Clc1ccc2c(c1)N=C1C3CCC(C3)CN1C2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 3/20 0.44
CTSD P07339 6/20 0.39
PDE3B Q13370 1/20 0.33
PDE3A Q14432 1/20 0.33
BCHE P06276 2/20 0.33
HRH4 Q9H3N8 3/20 0.31
CCR3 P51677 1/20 0.31
DRD2 P14416 2/20 0.30
DRD4 P21917 2/20 0.30
KCNK2 O95069 1/20 0.30
ADRB2 P07550 1/20 0.30
CHRM2 P08172 1/20 0.30
CHRM4 P08173 1/20 0.30
HTR1A P08908 1/20 0.30
CHRM5 P08912 1/20 0.30
ADRA2A P08913 1/20 0.30
ADORA3 P0DMS8 1/20 0.30
CHRM1 P11229 1/20 0.30
ADRA2B P18089 1/20 0.30
ADRA2C P18825 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8969872 0.80
SCHEMBL8969410 0.76 NOS1 (0.30)
SCHEMBL8969499 0.76 CTSD (0.49) ACHECTSDHRH4HTR2AHTR2C
SCHEMBL8968819 0.74 MAPK1 (0.34) ACHEBCHEHRH4CCR3CHRM1
SCHEMBL8969540 0.74 BCHE (0.32) ACHEBCHE
SCHEMBL8969466 0.73 CTSD (0.49) ACHECTSDHTR2AHTR2CHTR2B
SCHEMBL8968679 0.71 CTSD (0.47) ACHECTSDHTR2AHTR2CHRH1
SCHEMBL8968807 0.70
SCHEMBL24331504 0.68 ACHE (0.46) ACHECTSDPDE3BPDE3AHRH4
SCHEMBL8969755 0.66 EGFR (0.35) ACHEPDE3BPDE3ABCHEHRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5486512-A LEARNING ENHANCEMENT WARNER-LAMBERT COMPANY (US) 1996-01-23 US disclosed
EP-0597956-A1 QUINAZOLINE DERIVATIVES AS ACETYLCHOLINESTERASE INHIBITORS WARNER-LAMBERT COMPANY (US) 1994-05-25 EP disclosed
WO-1993003034-A1 QUINAZOLINE DERIVATIVES AS ACETYLCHOLINESTERASE INHIBITORS WARNER-LAMBERT COMPANY (US) 1993-02-18 WO disclosed