SCHEMBL8970277

SCHEMBL8970277

COc1cccc2c1CC(CNCCCCn1cccc/c1=N\S(C)(=O)=O)CC2

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.43
CHRM1 P11229 1/20 0.43
CHRM3 P20309 1/20 0.43
MTNR1A P48039 7/20 0.41
MTNR1B P49286 7/20 0.41
HTR1A P08908 2/20 0.40
SIGMAR1 Q99720 1/20 0.40
DRD2 P14416 1/20 0.40
DRD1 P21728 1/20 0.40
HTR1B P28222 1/20 0.40
HTR2A P28223 1/20 0.40
CYP1A2 P05177 1/20 0.39
MAPT P10636 1/20 0.39
CYP2C9 P11712 1/20 0.39
ALOX15 P16050 1/20 0.39
ADRA1D P25100 1/20 0.39
ADRA1A P35348 1/20 0.39
ADRA1B P35368 1/20 0.39
EPHX2 P34913 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8970281 1.00 CHRM2 (0.43) CHRM2CHRM1CHRM3MTNR1AMTNR1B
SCHEMBL9382674 0.76 CHRM2 (0.45) CHRM2CHRM1CHRM3MTNR1AMTNR1B
SCHEMBL9382677 0.74 ADRA1D (0.42) CHRM2CHRM1CHRM3MTNR1AMTNR1B
SCHEMBL8969041 0.73 CHRM2 (0.51) CHRM2CHRM1CHRM3MTNR1AMTNR1B
SCHEMBL8970407 0.73 SIGMAR1 (0.53) CHRM2CHRM1CHRM3MTNR1AMTNR1B
SCHEMBL8971218 0.73 HTR1A (0.59) HTR1ADRD2HTR2A
SCHEMBL8996726 0.73 HTR1A (0.49) CHRM2CHRM1CHRM3MTNR1AMTNR1B
SCHEMBL8970496 0.73 CHRM2 (0.48) CHRM2CHRM1CHRM3MTNR1AMTNR1B
SCHEMBL8969531 0.72 HTR7 (0.55) CHRM2CHRM1CHRM3HTR1ADRD2
SCHEMBL8970307 0.72 MTNR1A (0.62) CHRM2CHRM1CHRM3MTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5585392-A TREATING OR PREVENTING STROKES BAYER AKTIENGESELLSCHAFT (DE) 1996-12-17 US disclosed
US-5506246-A Method for treating depression using substituted aminomethyltetralins and their heterocyclic analogues BAYER AKTIENGESELLSCHAFT (DE) 1996-04-09 US disclosed
US-5300523-A Binding serotonin receptors, treating nervous system disorders BAYER AKTIENGESELLSCHAFT (DE) 1994-04-05 US disclosed
US-5137901-A For binding 5-HT 1 receptors; treating central nervous system disorders BAYER AKTIENGESELLSCHAFT (DE) 1992-08-11 US disclosed