SCHEMBL9687922

SCHEMBL9687922

CCn1c(C(=O)O)cc2cc(NC(=O)OCc3ccccc3)ccc21.O=C(Nc1ccc2[nH]c(C(=O)O)cc2c1)OCc1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 3/20 0.46
ALDH1A1 P00352 2/20 0.46
KDM4E B2RXH2 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2C9 P11712 1/20 0.46
HPGD P15428 1/20 0.46
HSD17B10 Q99714 1/20 0.46
ROCK2 O75116 2/20 0.44
MMP13 P45452 1/20 0.42
MGLL Q99685 2/20 0.41
SRD5A1 P18405 1/20 0.41
NPC1 O15118 1/20 0.40
TP53 P04637 1/20 0.40
MAPT P10636 1/20 0.40
TSHR P16473 1/20 0.40
RAB9A P51151 1/20 0.40
ATM Q13315 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
ADORA2B P29275 2/20 0.39
ADORA3 P0DMS8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9687928 0.90 MMP13 (0.46) SRD5A2ALDH1A1KDM4ECYP1A2CYP2C9
SCHEMBL8985906 0.86 SRD5A2 (0.60) SRD5A2ALDH1A1KDM4ECYP1A2CYP2C9
SCHEMBL8985820 0.79 MMP13 (0.68) ALDH1A1KDM4EHPGDHSD17B10ROCK2
SCHEMBL9688119 0.74 MMP13 (0.61) ALDH1A1KDM4EHPGDHSD17B10ROCK2
SCHEMBL5200855 0.72 MGLL (0.60) ALDH1A1ROCK2MGLLNPC1TP53
SCHEMBL7833243 0.71 LEF1 (0.55) SRD5A2ALDH1A1KDM4ECYP1A2CYP2C9
SCHEMBL7908588 0.70 KCNQ2 (0.57) ALDH1A1ROCK2MGLLNPC1TP53
SCHEMBL28292646 0.70 SERPINE1 (0.45) ALDH1A1HPGDROCK2TP53MAPT
SCHEMBL9127299 0.70 NPC1 (0.67) ALDH1A1KDM4ENPC1RAB9ASMN1; SMN2
SCHEMBL700511 0.70 SRD5A2 (0.73) SRD5A2ALDH1A1KDM4ECYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0507861-A1 DIAROMATIC SUBSTITUTED ANTI-AIDS COMPOUNDS. UPJOHN CO (US) 1992-10-14 EP disclosed
WO-1991009849-A1 DIAROMATIC SUBSTITUTED ANTI-AIDS COMPOUNDS THE UPJOHN COMPANY (US) 1991-07-11 WO disclosed