SCHEMBL898781

SCHEMBL898781

Fc1cc(-c2cn(Cc3ccccc3)c(=Nc3ccccc3)s2)ccn1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 3/20 0.41
ROCK1 Q13464 3/20 0.41
EGLN1 Q9GZT9 1/20 0.35
PDE4D Q08499 1/20 0.34
PDE7A Q13946 1/20 0.34
KDM5B Q9UGL1 1/20 0.34
MAPK1 P28482 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
MAPK14 Q16539 3/20 0.33
GRM5 P41594 1/20 0.33
MAPK13 O15264 1/20 0.33
MAPK12 P53778 1/20 0.33
MAPK11 Q15759 1/20 0.33
CCNC P24863 1/20 0.33
CDK8 P49336 1/20 0.33
HTR6 P50406 1/20 0.32
KCNH2 Q12809 1/20 0.32
DYRK1A Q13627 1/20 0.32
CTSA P10619 1/20 0.31
LMNA P02545 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL898780 1.00 ROCK2 (0.41) ROCK2ROCK1EGLN1PDE4DPDE7A
SCHEMBL899436 0.81 PDE4D (0.39) PDE4DPDE7AMAPK1NPSR1LMNA
SCHEMBL899437 0.81 PDE4D (0.39) PDE4DPDE7AMAPK1NPSR1LMNA
SCHEMBL899584 0.81 SMN1; SMN2 (0.42) PDE4DPDE7AMAPK1NPSR1LMNA
SCHEMBL899582 0.81 SMN1; SMN2 (0.42) PDE4DPDE7AMAPK1NPSR1LMNA
SCHEMBL898805 0.78 GRM5 (0.34) PDE4DPDE7AMAPK1NPSR1GRM5
SCHEMBL898806 0.78 GRM5 (0.34) PDE4DPDE7AMAPK1NPSR1GRM5
SCHEMBL899463 0.76 LMNA (0.43) MAPK1LMNAPOLBSMN1; SMN2RAB9A
SCHEMBL899307 0.73 MAPT (0.46) MAPK1NPSR1LMNASMN1; SMN2NPC1
SCHEMBL899306 0.73 MAPT (0.46) MAPK1NPSR1LMNASMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012040754-A2 NOVEL THIAZOLAMINE DERIVATES AS DIFFERENTIATION ACCELERATORS TECHNISCHE UNIVERSITÄT WIEN (AT) 2012-04-05 WO claimed
WO-2012040754-A2 NOVEL THIAZOLAMINE DERIVATES AS DIFFERENTIATION ACCELERATORS TECHNISCHE UNIVERSITÄT WIEN (AT) 2012-04-05 WO disclosed