SCHEMBL898826

SCHEMBL898826

O=[N+]([O-])c1ccc(-c2cnc(N(Cc3ccccc3)c3ccccc3)s2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
XDH P47989 1/20 0.48
CRHBP P24387 3/20 0.46
CRHR2 Q13324 3/20 0.46
AR P10275 5/20 0.43
APP P05067 2/20 0.41
MAPT P10636 2/20 0.41
CYP1A2 P05177 1/20 0.41
POLB P06746 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
ALDH1A1 P00352 4/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
LMNA P02545 2/20 0.40
ATM Q13315 1/20 0.40
TLR9 Q9NR96 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
KDM4E B2RXH2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL899467 0.90 ALDH1A1 (0.44) MAPTCYP1A2CYP2C9ALDH1A1LMNA
SCHEMBL899302 0.85 CCNE1 (0.42) ALDH1A1LMNAKDM4E
SCHEMBL899084 0.82 KCNH2 (0.38) MAPTNPSR1ALDH1A1L3MBTL1LMNA
SCHEMBL899508 0.82 HDAC1 (0.47) MAPTCYP3A4CYP2C9ALDH1A1MEN1
SCHEMBL903025 0.81 HDAC1 (0.40) CYP3A4ALDH1A1KDM4E
SCHEMBL899366 0.79 HSD17B2 (0.46) APPLMNASMN1; SMN2MMP2MMP9
SCHEMBL902944 0.77 HDAC1 (0.38) ALDH1A1KDM4E
SCHEMBL5843018 0.77 CRHBP (0.64) CRHBPCRHR2ARCYP1A2CYP2C9
SCHEMBL20379759 0.74 XDH (0.76) XDHAPPMAPTPOLBCYP3A4
SCHEMBL899484 0.73 ALDH1A1 (0.38) MAPTCYP1A2POLBCYP2C9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012040754-A2 NOVEL THIAZOLAMINE DERIVATES AS DIFFERENTIATION ACCELERATORS TECHNISCHE UNIVERSITÄT WIEN (AT) 2012-04-05 WO disclosed
WO-2012040754-A2 NOVEL THIAZOLAMINE DERIVATES AS DIFFERENTIATION ACCELERATORS TECHNISCHE UNIVERSITÄT WIEN (AT) 2012-04-05 WO disclosed