SCHEMBL8993148

SCHEMBL8993148

COc1cc(Cc2ccc(-c3cnn4c(O)ncnc34)cc2)cc(OC)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
CALM1 P0DP23 2/20 0.40
MAPT P10636 4/20 0.38
KDR P35968 4/20 0.38
LMNA P02545 1/20 0.38
MEN1 O00255 2/20 0.38
MAPK1 P28482 1/20 0.38
STAT1 P42224 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
HCAR2 Q8TDS4 2/20 0.37
HPGD P15428 1/20 0.36
PDE1B Q01064 1/20 0.35
TP53 P04637 1/20 0.35
BMP4 P12644 1/20 0.34
FLT1 P17948 1/20 0.34
FLT4 P35916 1/20 0.34
EGLN1 Q9GZT9 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8992990 0.92 KMT2A (0.48) KMT2ANPC1RAB9AMAPTKDR
SCHEMBL8992950 0.90 LTA4H (0.43) KMT2ANPC1RAB9AMAPTLMNA
SCHEMBL9217924 0.84 KMT2A (0.54) KMT2ANPC1RAB9AMAPTKDR
SCHEMBL9215969 0.84 CYP1A1 (0.42) KMT2ANPC1RAB9AMAPTKDR
SCHEMBL8992965 0.83 GPR119 (0.41) KMT2ANPC1RAB9AMAPTKDR
SCHEMBL8993293 0.82 KMT2A (0.40) KMT2ANPC1RAB9AMAPTKDR
SCHEMBL8992955 0.82 NPC1 (0.43) KMT2ANPC1RAB9AMAPTMEN1
SCHEMBL8993213 0.81 RAB9A (0.46) KMT2ANPC1RAB9AMAPTKDR
SCHEMBL8992831 0.80 LTA4H (0.42) KMT2ANPC1RAB9AMAPTLMNA
SCHEMBL8992922 0.80 GPR119 (0.43) KMT2ANPC1RAB9AKDRMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5516777-A PROSTATE CANCER THERAPY OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1996-05-14 US disclosed
US-5409928-A Prostate diseases, alopecia OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-04-25 US disclosed
EP-0594149-A2 Condensed pyrazole derivatives, method of manufacturing the same, and androgen inhibitor OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-04-27 EP disclosed