SCHEMBL899483

SCHEMBL899483

Cc1ccc(N=c2sc(-c3cccnc3F)cn2Cc2ccccc2)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.36
SMN1; SMN2 Q16637 5/20 0.34
NPC1 O15118 5/20 0.34
RAB9A P51151 5/20 0.34
LMNA P02545 4/20 0.34
ALDH1A1 P00352 3/20 0.34
POLB P06746 3/20 0.34
L3MBTL1 Q9Y468 3/20 0.34
KDM4E B2RXH2 2/20 0.34
MAPT P10636 2/20 0.34
S1PR2 O95136 1/20 0.34
GLA P06280 1/20 0.34
GAA P10253 1/20 0.34
HPGD P15428 1/20 0.34
ATM Q13315 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
CA9 Q16790 1/20 0.33
CYP11B1 P15538 1/20 0.32
CYP11B2 P19099 1/20 0.32
HTT P42858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL898806 0.92 GRM5 (0.34) SMN1; SMN2NPC1RAB9AALDH1A1L3MBTL1
SCHEMBL898805 0.92 GRM5 (0.34) SMN1; SMN2NPC1RAB9AALDH1A1L3MBTL1
SCHEMBL899322 0.85 OPRD1 (0.35) SMN1; SMN2NPC1RAB9ALMNAALDH1A1
SCHEMBL899220 0.77 PDE4D (0.38) PTGS2SMN1; SMN2NPC1RAB9AALDH1A1
SCHEMBL899381 0.77 MAPT (0.41) PTGS2SMN1; SMN2NPC1RAB9ALMNA
SCHEMBL899380 0.77 MAPT (0.41) PTGS2SMN1; SMN2NPC1RAB9ALMNA
SCHEMBL898781 0.72 ROCK2 (0.41) SMN1; SMN2NPC1RAB9ALMNAPOLB
SCHEMBL898780 0.72 ROCK2 (0.41) SMN1; SMN2NPC1RAB9ALMNAPOLB
SCHEMBL899437 0.70 PDE4D (0.39) SMN1; SMN2NPC1RAB9ALMNAALDH1A1
SCHEMBL899436 0.70 PDE4D (0.39) SMN1; SMN2NPC1RAB9ALMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012040754-A2 NOVEL THIAZOLAMINE DERIVATES AS DIFFERENTIATION ACCELERATORS TECHNISCHE UNIVERSITÄT WIEN (AT) 2012-04-05 WO disclosed