SCHEMBL8997603

SCHEMBL8997603

CCN(C[C@H](C)COc1cccc2c1C[C@](NC(=O)OC(C)(C)C)(OC(=O)OC)CC2)C(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)OCc1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SYK P43405 1/20 0.38
CTSK P43235 4/20 0.34
CTSL P07711 2/20 0.33
CTSS P25774 2/20 0.33
CTSB P07858 1/20 0.33
PSEN1 P49768 2/20 0.33
PSEN2 P49810 2/20 0.33
APH1B Q8WW43 2/20 0.33
NCSTN Q92542 2/20 0.33
APH1A Q96BI3 2/20 0.33
PSENEN Q9NZ42 2/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
ACHE P22303 1/20 0.33
PSMB5 P28074 2/20 0.32
CYP1A2 P05177 2/20 0.32
MEN1 O00255 2/20 0.32
LMNA P02545 2/20 0.32
KMT2A Q03164 2/20 0.32
GHSR Q92847 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8997612 0.89 SYK (0.41) SYKCTSKCTSBCA1CA2
SCHEMBL8997623 0.88 GHSR (0.34) GHSR
SCHEMBL8997761 0.85 GHSR (0.33) GHSR
SCHEMBL8997594 0.80 SYK (0.40) SYKCTSKCA1CA2ACHE
SCHEMBL8582293 0.78 SYK (0.44) SYKCTSKCTSLCTSSCTSB
SCHEMBL8997804 0.78 P2RY1 (0.37) SYKCTSKCYP1A2CYP3A4CYP2C9
SCHEMBL8997619 0.78 GHSR (0.35) CYP1A2LMNAGHSRCYP2C9TSHR
SCHEMBL8997596 0.77 GHSR (0.35) LMNAGHSRTSHR
SCHEMBL8997607 0.77 GHSR (0.35) CYP1A2LMNAGHSRCYP2C9TSHR
SCHEMBL8997600 0.76 SYK (0.40) SYKCA1CA2ACHECYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0729972-A1 Peptide derivatives of tetrahydronaphthalene F. HOFFMANN-LA ROCHE AG (CH) 1996-09-04 EP disclosed