SCHEMBL8997612

SCHEMBL8997612

COC(=O)O[C@]1(NC(=O)OC(C)(C)C)CCc2cccc(OC[C@@H](C)CNC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)OCc3ccccc3)c2C1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SYK P43405 1/20 0.41
CYP1A2 P05177 4/20 0.37
CTSK P43235 1/20 0.36
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
ACHE P22303 1/20 0.34
PSMB5 P28074 2/20 0.34
LGMN Q99538 1/20 0.34
TPSAB1 Q15661 2/20 0.33
PLG P00747 1/20 0.33
PRSS1 P07477 1/20 0.33
CTSB P07858 1/20 0.33
NTSR1 P30989 1/20 0.33
CYP3A4 P08684 3/20 0.33
CYP2D6 P10635 3/20 0.33
CYP2C9 P11712 3/20 0.33
CYP2C19 P33261 3/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
ALDH1A1 P00352 1/20 0.33
TSHR P16473 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8997603 0.89 SYK (0.38) SYKCYP1A2CTSKCA1CA2
SCHEMBL8582293 0.89 SYK (0.44) SYKCYP1A2CTSKCA1CA2
SCHEMBL8997886 0.86 PRMT5 (0.31)
SCHEMBL8997715 0.84 CPB2 (0.31)
SCHEMBL8997594 0.83 SYK (0.40) SYKCYP1A2CTSKCA1CA2
SCHEMBL8997804 0.81 P2RY1 (0.37) SYKCYP1A2CTSKCYP3A4CYP2D6
SCHEMBL8997607 0.81 GHSR (0.35) CYP1A2CYP2C9TSHR
SCHEMBL8997619 0.80 GHSR (0.35) CYP1A2CYP2C9TSHR
SCHEMBL8997596 0.80 GHSR (0.35) TSHR
SCHEMBL8997593 0.79 ALDH1A1 (0.35) SYKCYP1A2CA1CA2ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0729972-A1 Peptide derivatives of tetrahydronaphthalene F. HOFFMANN-LA ROCHE AG (CH) 1996-09-04 EP disclosed