SCHEMBL8997631

SCHEMBL8997631

C[C@H](N)C(=O)Nc1ccccc1Oc1cccc2c1C[C@](NC(=O)OC(C)(C)C)(OC(=O)OCc1ccccc1)CC2

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SYK P43405 1/20 0.35
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
ACHE P22303 1/20 0.34
GHSR Q92847 1/20 0.34
LTA4H P09960 1/20 0.33
PRMT5 O14744 1/20 0.33
WDR77 Q9BQA1 1/20 0.33
BRD4 O60885 1/20 0.32
CASP3 P42574 1/20 0.32
XIAP P98170 1/20 0.32
AAK1 Q2M2I8 1/20 0.31
PSMB5 P28074 1/20 0.31
CTSK P43235 2/20 0.31
CARM1 Q86X55 1/20 0.31
IDO1 P14902 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8997810 0.92 P2RY1 (0.39)
SCHEMBL8997594 0.90 SYK (0.40) SYKCA1CA2ACHEPSMB5
SCHEMBL8997648 0.86 SYK (0.38) SYKCA1CA2ACHEGHSR
SCHEMBL8997716 0.85 GHSR (0.33) GHSRPRMT5WDR77CASP3IDO1
SCHEMBL8997804 0.83 P2RY1 (0.37) SYKCTSK
SCHEMBL8567143 0.82 CA1 (0.39) SYKCA1CA2ACHEGHSR
SCHEMBL8575729 0.82 CA1 (0.39) SYKCA1CA2ACHEGHSR
SCHEMBL8997699 0.82 CA1 (0.36) SYKCA1CA2ACHEGHSR
SCHEMBL8997628 0.81 CA1 (0.34) SYKCA1CA2ACHEGHSR
SCHEMBL8561322 0.81 SYK (0.40) SYKCA1CA2ACHEGHSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0729972-A1 Peptide derivatives of tetrahydronaphthalene F. HOFFMANN-LA ROCHE AG (CH) 1996-09-04 EP disclosed