SCHEMBL9001876

SCHEMBL9001876

O=C(NCCSc1cccc2nccn12)OCC1c2ccccc2-c2ccccc21

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.47
EPHX2 P34913 1/20 0.41
DOT1L Q8TEK3 1/20 0.38
MDM4 O15151 1/20 0.36
TP53 P04637 1/20 0.36
OPRD1 P41143 1/20 0.35
HDAC1 Q13547 1/20 0.34
HDAC2 Q92769 1/20 0.34
CASP3 P42574 1/20 0.34
FABP7 O15540 1/20 0.33
FABP5 Q01469 1/20 0.33
CXCR2 P25025 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9001977 0.80 MTNR1B (0.37) KMT2ATP53
SCHEMBL9001857 0.80 HPGD (0.34) EPHX2TP53
SCHEMBL9002020 0.79 CASP1 (0.33) KMT2A
SCHEMBL9001916 0.77 SMN1; SMN2 (0.36) KMT2ATP53
SCHEMBL9002320 0.77 BRD4 (0.42)
Hydrochloric Acid SCHEMBL9001979 0.76 SMN1; SMN2 (0.36) KMT2ATP53
SCHEMBL9001920 0.76 MTNR1A (0.47) KMT2A
SCHEMBL9001895 0.73 ACHE (0.38) EPHX2
SCHEMBL9001872 0.73 CDK8 (0.34) KMT2A
SCHEMBL9002205 0.73 ALDH1A1 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5587383-A CALMODULIN INHIBITORS; ANTIISCHEMIC AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-12-24 US disclosed
EP-0471236-B1 Imidazopyridine derivatives and their use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1995-03-15 EP disclosed
US-5395839-A Calmodulin and angiogenesis inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-03-07 US disclosed
US-5244908-A Calmodulin inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-09-14 US disclosed
EP-0471236-A1 Imidazopyridine derivatives and their use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-02-19 EP disclosed