SCHEMBL9006005

SCHEMBL9006005

Nc1c(CP(=O)(O)O)c(CCC(=O)O)nc2cc(Cl)ccc12

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
KMT2A Q03164 1/20 0.43
HDAC6 Q9UBN7 1/20 0.42
GPR17 Q13304 1/20 0.39
FFAR1 O14842 1/20 0.38
ACHE P22303 3/20 0.36
BCHE P06276 2/20 0.36
CHRM1 P11229 1/20 0.36
EPHX2 P34913 1/20 0.36
NR4A2 P43354 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9005979 0.81 KDM4E (0.36) KDM4EHDAC6
SCHEMBL9005993 0.70 KDM4E (0.42) KDM4EALDH1A1HDAC6
SCHEMBL8936196 0.68 IGFBP5 (0.43) KMT2A
SCHEMBL9700784 0.64 HDAC6 (0.41) KDM4EALDH1A1HDAC6CHRM1
SCHEMBL9700703 0.64
SCHEMBL8708279 0.63 TBXA2R (0.54) KDM4EALDH1A1HDAC6
SCHEMBL8645093 0.63 PRKAG1 (0.37)
SCHEMBL8614149 0.63 HDAC6 (0.70) KDM4EALDH1A1KMT2AHDAC6
SCHEMBL3362000 0.63 APP (0.46) KDM4EALDH1A1KMT2AACHEBCHE
SCHEMBL8644010 0.62

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0736032-A1 HETEROCYCLIC COMPOUNDS Astra Aktiebolag (SE) 1996-10-09 EP disclosed
WO-1995017410-A1 HETEROCYCLIC COMPOUNDS ASTRA AKTIEBOLAG (SE) 1995-06-29 WO disclosed