SCHEMBL901345

SCHEMBL901345

O=C(O)C1CC2CCN1C2

nearest known ligand 0.37

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.35
ACE P12821 5/20 0.34
AGTR2 P50052 2/20 0.32
ALDH1A1 P00352 2/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
REN P00797 1/20 0.32
NOTUM Q6P988 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2428126 1.00 ATM (0.35) ATMACEAGTR2ALDH1A1SMN1; SMN2
SCHEMBL15265282 0.90 ALDH1A1 (0.42) ACEALDH1A1SMN1; SMN2REN
SCHEMBL572684 0.86 ACE (0.36) ATMACEALDH1A1SMN1; SMN2
SCHEMBL357830 0.84 ATM (0.34) ATMACEAGTR2ALDH1A1SMN1; SMN2
SCHEMBL4024975 0.84
Hydrochloric Acid SCHEMBL14343221 0.84 ACE (0.35) ATMACEALDH1A1SMN1; SMN2
Hydrochloric Acid SCHEMBL14343353 0.84 ACE (0.35) ATMACEALDH1A1SMN1; SMN2
Bromide SCHEMBL28148076 0.84 ACE (0.35) ATMACEALDH1A1SMN1; SMN2
Hydrochloric Acid SCHEMBL5473763 0.84 ACE (0.35) ATMACEALDH1A1SMN1; SMN2
SCHEMBL30369975 0.83

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 64 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240239792-A1 MODULATORS OF BCL-2 OR BCL-2/BCL-XL AND USES THEREOF ASIA VISION LIMITED (CN) 2024-07-18 US claimed
WO-2025233863-A1 ENPP1 INHIBITORS RE VENTURES I, LLC (US) 2025-11-13 WO disclosed
US-20240239792-A1 MODULATORS OF BCL-2 OR BCL-2/BCL-XL AND USES THEREOF ASIA VISION LIMITED (CN) 2024-07-18 US disclosed
US-11964989-B2 KRas G12D inhibitors Mirati Therapeutics, Inc. (US) 2024-04-23 US disclosed
US-20240025920-A1 SALT FORM USED AS CDC7 INHIBITOR AND CRYSTAL FORM THEREOF CHIA TAI TIANQING PHARMACEUTICAL GROUP CO., LTD. (CN) 2024-01-25 US disclosed
US-20240025920-A1 SALT FORM USED AS CDC7 INHIBITOR AND CRYSTAL FORM THEREOF CHIA TAI TIANQING PHARMACEUTICAL GROUP CO., LTD. (CN) 2024-01-25 US disclosed
EP-4277895-A1 HETEROCYCLIC P2Y 14 RECEPTOR ANTAGONISTS The United States of America, as represented by the Secretary, Department of Health and Human Services (US) 2023-11-22 EP disclosed
EP-4253388-A1 SALT FORM USED AS CDC7 INHIBITOR AND CRYSTAL FORM THEREOF CHIA TAI TIANQING PHARMACEUTICAL GROUP CO., LTD. (CN) 2023-10-04 EP disclosed
US-20230077225-A1 KRAS G12D INHIBITORS Mirati Therapeutics, Inc. 2023-03-09 US disclosed
WO-2022155037-A1 HETEROCYCLIC P2Y 14 RECEPTOR ANTAGONISTS THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2022-07-21 WO disclosed
US-20060217406-A1 N-ARYL DIAZASPIRACYCLIC COMPOUNDS AND METHODS OF PREPARATION AND USE THEREOF BHATTI BALWINDER S 2006-09-28 US disclosed
US-20060058328-A1 Use of N-aryl diazaspiracyclic compounds in the treatment of addiction BHATTI BALWINDER S 2006-03-16 US disclosed
WO-2006023630-A2 THE USE OF N-ARYL DIAZASPIRACYCLIC COMPOUNDS IN THE TREATMENT OF ADDICTION TARGACEPT, INC. (US) 2006-03-02 WO disclosed
US-20050272739-A1 N-aryl diazaspiracyclic compounds and methods of preparation and use thereof BHATTI BALWINDER S 2005-12-08 US disclosed
US-6956042-B2 N-aryl diazaspiracyclic compounds and methods of preparation and use thereof TARGACEPT, INC. (US) 2005-10-18 US disclosed
WO-2005042533-A2 2-CYANOPYRROLIDINECARBOXAMIDES AS DIPEPTIDYL PEPTIDASE-IV INHIBITORS ASTELLAS PHARMA INC. (JP) 2005-05-12 WO disclosed
EP-1519939-A2 N-ARYL DIAZASPIRACYCLIC COMPOUNDS AND METHODS OF PREPARATION AND USE THEREOF Targacept, Inc. (US) 2005-04-06 EP disclosed
US-20040067930-A1 N-aryl diazaspiracyclic compounds and methods of preparation and use thereof TARGACEPT, INC. 2004-04-08 US disclosed
WO-2004009599-A1 FIVE-MEMBERED HETEROAROMATIC OLEFINIC AZACYCLIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR USE AS INHIBITORS OF NCOTINIC CHOLINERGIC RECEPTORS TARGACEPT, INC. (US) 2004-01-29 WO disclosed
WO-2004005293-A2 N-ARYL DIAZASPIRACYCLIC COMPOUNDS AND METHODS OF PREPARATION AND USE THEREOF TARGACEPT, INC. (US) 2004-01-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240239792-A1 MODULATORS OF BCL-2 OR BCL-2/BCL-XL AND USES THEREOF BCL2, BCL2L2, BCL2L1 ATM 3016/4885ACE 4562/4885AGTR2 2249/4885
US-20230077225-A1 KRAS G12D INHIBITORS KRAS, NRAS, HRAS ATM 3658/4885ACE 1101/4885AGTR2 1496/4885
US-20240025920-A1 SALT FORM USED AS CDC7 INHIBITOR AND CRYSTAL FORM THEREOF CDC7, CDC73, CDC5L ATM 1882/4885ACE 772/4885AGTR2 2449/4885
US-20060217406-A1 N-ARYL DIAZASPIRACYCLIC COMPOUNDS AND METHODS OF PREPARATION AND USE THEREOF TNNC1, ACHE, CHRNA6 ATM 3528/4885ACE 701/4885AGTR2 252/4885
US-11964989-B2 KRas G12D inhibitors KRAS, NRAS, HRAS ATM 3241/4885ACE 532/4885AGTR2 749/4885
US-20050272739-A1 N-aryl diazaspiracyclic compounds and methods of preparation and use thereof TNNC1, ACHE, CHRNA6 ATM 3528/4885ACE 701/4885AGTR2 252/4885
US-20060058328-A1 Use of N-aryl diazaspiracyclic compounds in the treatment of addiction OPRD1, OPRK1, OPRL1 ATM 1307/4885ACE 220/4885AGTR2 153/4885
US-20040067930-A1 N-aryl diazaspiracyclic compounds and methods of preparation and use thereof TNNC1, ACHE, CHRNA6 ATM 3528/4885ACE 701/4885AGTR2 252/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.