SCHEMBL9014302

SCHEMBL9014302

COc1ccc2c(c1)C(CCBr)CCCO2

nearest known ligand 0.60

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 4/20 0.47
ENPP2 Q13822 1/20 0.42
SIGMAR1 Q99720 3/20 0.41
HTR2B P41595 2/20 0.41
HTR7 P34969 1/20 0.41
TMEM97 Q5BJF2 1/20 0.41
MTNR1A P48039 6/20 0.40
MTNR1B P49286 5/20 0.40
NQO2 P16083 3/20 0.38
DRD2 P14416 1/20 0.37
DRD3 P35462 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10407585 0.92 HTR1A (0.54) HTR1AENPP2SIGMAR1HTR2BHTR7
SCHEMBL9014335 0.80 KDM4E (0.37) HTR1AMTNR1AMTNR1B
SCHEMBL9234439 0.80 DRD3 (0.37) HTR1ADRD2DRD3
SCHEMBL9014788 0.80 ADRA2A (0.40) HTR1AMTNR1AMTNR1BDRD2DRD3
SCHEMBL5479142 0.78 HTR1A (0.54) HTR1AENPP2SIGMAR1HTR2BHTR7
SCHEMBL9014733 0.76 DRD2 (0.39) DRD2DRD3
SCHEMBL9014727 0.76 KCNH2 (0.38) MTNR1AMTNR1B
SCHEMBL9014779 0.73 KCNH2 (0.70) ENPP2SIGMAR1DRD2
SCHEMBL7950300 0.73 MTNR1A (0.62) MTNR1AMTNR1BNQO2
SCHEMBL24915792 0.73 ENPP2 (0.48) HTR1AENPP2SIGMAR1HTR2BHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5495022-A Piperidines and piperazines MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1996-02-27 US disclosed
EP-0634398-A1 4-Phenylpiperidinyl-1/-piperazinyl-1-ethylsubstituted benzofusedheterocycles as antiarrhythmic agents MERCK PATENT GmbH (DE) 1995-01-18 EP disclosed