SCHEMBL9014357

SCHEMBL9014357

CCC(=O)N1CCC(CCN2CCC(c3ccc(Cl)cc3)CC2)c2ccccc21

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 7/20 0.54
MCHR1 Q99705 3/20 0.45
PRCP P42785 5/20 0.44
DRD4 P21917 2/20 0.42
DRD3 P35462 2/20 0.42
SLC6A4 P31645 1/20 0.41
CCR1 P32246 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
SIGMAR1 Q99720 2/20 0.41
KCNH2 Q12809 1/20 0.41
CHRM4 P08173 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9014749 0.92 DRD2 (0.53) DRD2PRCPSIGMAR1
SCHEMBL9014672 0.88 DRD2 (0.55) DRD2DRD3SIGMAR1KCNH2CHRM4
SCHEMBL9014708 0.84 KCNH2 (0.61) DRD2SLC6A4MEN1KMT2AKCNH2
SCHEMBL9014782 0.84 KCNH2 (0.47) DRD2DRD3SLC6A4KCNH2
SCHEMBL9014707 0.79 DRD2 (0.52) DRD2PRCPDRD4DRD3MEN1
SCHEMBL9014839 0.78 DRD2 (0.54) DRD2SIGMAR1KCNH2CHRM4
SCHEMBL11839176 0.75 DRD2 (0.57) DRD2PRCPKMT2ASIGMAR1
SCHEMBL6790341 0.75 DRD2 (0.55) DRD2MCHR1DRD4DRD3SIGMAR1
SCHEMBL6792592 0.74 DRD2 (0.52) DRD2MCHR1DRD4SLC6A4MEN1
SCHEMBL9014725 0.73 KCNH2 (0.63) DRD2DRD4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5495022-A Piperidines and piperazines MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1996-02-27 US disclosed
EP-0634398-A1 4-Phenylpiperidinyl-1/-piperazinyl-1-ethylsubstituted benzofusedheterocycles as antiarrhythmic agents MERCK PATENT GmbH (DE) 1995-01-18 EP disclosed